Suchergebnisse - "Brewitz, Lennart"

PubPharm (49)

1

Studies on the selectivity of the SARS-CoV-2 papain-like protease reveal the importance of the P2′ proline of the viral polyprotein

enthalten in: bioRxiv.org | 2024

von Chan, H. | Brewitz, L. | Lukacik, P. | +4

2

The selective prolyl hydroxylase inhibitor IOX5 stabilizes HIF-1α and compromises development and progression of acute myeloid leukemia

enthalten in: Nature cancer | 2024

von Lawson, H. | Holt-Martyn, J. | Dembitz, V. | +25

3

Studies on the selectivity of the SARS-CoV-2 papain-like protease reveal the importance of the P2' proline of the viral polyprotein

enthalten in: RSC chemical biology | 2024

von Chan, H. | Brewitz, L. | Lukacik, P. | +4

4

Mass spectrometric assays monitoring the deubiquitinase activity of the SARS-CoV-2 papain-like protease inform on the basis of substrate selectivity and have utility for substrate identification

enthalten in: Bioorganic & medicinal chemistry | 2023

von Brewitz, L. | Henry Chan, H. | Lukacik, P. | +4

5

Open science discovery of potent noncovalent SARS-CoV-2 main protease inhibitors

enthalten in: Science (New York, N.Y.) | 2023

von Boby, M. | Fearon, D. | Ferla, M. | +98

CommentIn: Nat Rev Drug Discov. 2024 Jan;23(1):22. - PMID 38040790

6

Structure-guided optimisation of N-hydroxythiazole-derived inhibitors of factor inhibiting hypoxia-inducible factor-α

enthalten in: Chemical science | 2023

von Corner, T. | Teo, R. | Wu, Y. | +10

7

αβ,α'β'-Diepoxyketones are mechanism-based inhibitors of nucleophilic cysteine enzymes

enthalten in: Chemical communications (Cambridge, England) | 2023

von de Munnik, M. | Lithgow, J. | Brewitz, L. | +4

8

5-Substituted Pyridine-2,4-dicarboxylate Derivatives Have Potential for Selective Inhibition of Human Jumonji-C Domain-Containing Protein 5

enthalten in: Journal of medicinal chemistry | 2023

von Brewitz, L. | Nakashima, Y. | Piasecka, S. | +10

9

In vitro selection of macrocyclic peptide inhibitors containing cyclic γ2,4-amino acids targeting the SARS-CoV-2 main protease

enthalten in: Nature chemistry | 2023

von Miura, T. | Malla, T. | Owen, C. | +13

10

Kinetic and inhibition studies on human Jumonji-C (JmjC) domain-containing protein 5

enthalten in: RSC chemical biology | 2023

von Tumber, A. | Salah, E. | Brewitz, L. | +2

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