Suchergebnisse - "Underwood, Elizabeth"

PubPharm (22)

1

Dynamics of the HD regulatory subdomain of PARP-1; substrate access and allostery in PARP activation and inhibition

enthalten in: bioRxiv.org | 2021

von Ogden, T. | Yang, J. | Schimpl, M. | +8

2

Discovery of 5-{4-[(7-Ethyl-6-oxo-5,6-dihydro-1,5-naphthyridin-3-yl)methyl]piperazin-1-yl}-N-methylpyridine-2-carboxamide (AZD5305) : A PARP1-DNA Trapper with High Selectivity for PARP1 over PARP2 and Other PARPs

enthalten in: Journal of medicinal chemistry | 2021

von Johannes, J. | Balazs, A. | Barratt, D. | +40

3

Fragment-Based Design of a Potent MAT2a Inhibitor and in Vivo Evaluation in an MTAP Null Xenograft Model

enthalten in: Journal of medicinal chemistry | 2021

von De Fusco, C. | Schimpl, M. | Börjesson, U. | +18

4

Generating Selective Leads for Mer Kinase Inhibitors-Example of a Comprehensive Lead-Generation Strategy

enthalten in: Journal of medicinal chemistry | 2021

von Nissink, J. | Bazzaz, S. | Blackett, C. | +26

5

Dynamics of the HD regulatory subdomain of PARP-1; substrate access and allostery in PARP activation and inhibition

enthalten in: Nucleic acids research | 2021

von Ogden, T. | Yang, J. | Schimpl, M. | +8

6

Characterization of the Kinetic Mechanism of Human Protein Arginine Methyltransferase 5

enthalten in: Biochemistry | 2020

von Eddershaw, A. | Stubbs, C. | Edwardes, L. | +5

7

A-loop interactions in Mer tyrosine kinase give rise to inhibitors with two-step mechanism and long residence time of binding

enthalten in: The Biochemical journal | 2020

von Pflug, A. | Schimpl, M. | Nissink, J. | +7

8

Effect of Phase II Match on residency program ranking of candidates

enthalten in: American journal of health-system pharmacy : AJHP : official journal of the American Society of Health-System Pharmacists | 2020

von Underwood, E. | Smith, M. | Hammond, D. | +1

9

Frequency of Occurrence of the Rat Lungworm Parasite in the Invasive Island Apple Snail in South Carolina, USA

enthalten in: Journal of aquatic animal health | 2019

von Underwood, E. | Walker, M. | Darden, T. | +1

10

Jarid2 binds mono-ubiquitylated H2A lysine 119 to mediate crosstalk between Polycomb complexes PRC1 and PRC2

enthalten in: Nature communications | 2016

von Cooper, S. | Grijzenhout, A. | Underwood, E. | +10