Suchergebnisse - "Song, Jen-Shin"

PubPharm (14)

1

Discovery and Synthesis of a Pyrimidine-Based Aurora Kinase Inhibitor to Reduce Levels of MYC Oncoproteins

enthalten in: Journal of medicinal chemistry | 2021

von Chi, Y. | Yeh, T. | Ke, Y. | +17

2

Drug-like property optimization : Discovery of orally bioavailable quinazoline-based multi-targeted kinase inhibitors

enthalten in: Bioorganic chemistry | 2020

von Lin, S. | Chang, C. | Coumar, M. | +14

3

Identification of a Multitargeted Tyrosine Kinase Inhibitor for the Treatment of Gastrointestinal Stromal Tumors and Acute Myeloid Leukemia

enthalten in: Journal of medicinal chemistry | 2019

von Lin, W. | Wu, S. | Yeh, T. | +25

4

Discovery of Conformational Control Inhibitors Switching off the Activated c-KIT and Targeting a Broad Range of Clinically Relevant c-KIT Mutants

enthalten in: Journal of medicinal chemistry | 2019

von Wu, T. | Lin, W. | Tsai, H. | +18

5

Design and synthesis of BPR1K653 derivatives targeting the back pocket of Aurora kinases for selective isoform inhibition

enthalten in: European journal of medicinal chemistry | 2018

von Ke, Y. | Chang, C. | Lin, W. | +12

6

Discovery of BPR1K871, a quinazoline based, multi-kinase inhibitor for the treatment of AML and solid tumors : Rational design, synthesis, in vitro and in vivo evaluation

enthalten in: Oncotarget | 2016

von Hsu, Y. | Coumar, M. | Wang, W. | +22

7

Synthesis of (E)-oxindolylidene acetate using tandem palladium-catalyzed Heck and alkoxycarbonylation reactions

enthalten in: Organic & biomolecular chemistry | 2016

von Lin, W. | Shia, K. | Song, J. | +2

8

Identification of a potent 5-phenyl-thiazol-2-ylamine-based inhibitor of FLT3 with activity against drug resistance-conferring point mutations

enthalten in: European journal of medicinal chemistry | 2015

von Chen, C. | Hsu, J. | Lin, W. | +15

9

Homology modeling of DFG-in FMS-like tyrosine kinase 3 (FLT3) and structure-based virtual screening for inhibitor identification

enthalten in: Scientific reports | 2015

von Ke, Y. | Singh, V. | Coumar, M. | +9

10

Ligand efficiency based approach for efficient virtual screening of compound libraries

enthalten in: European journal of medicinal chemistry | 2014

von Ke, Y. | Coumar, M. | Shiao, H. | +9