Suchergebnisse - "Lehmann, Jochen"

PubPharm (15)

1

Selective microemulsion liquid chromatography analysis of dopamine receptor antagonist LE300 and its N-methyl metabolite in mouse sera by using a monolithic silica column

enthalten in: Journal of chromatography. B, Analytical technologies in the biomedical and life sciences | 2015

von Al-Majed, A. | Hefnawy, M. | Mohammed, M. | +2

2

An interactive SAR approach to discover novel hybrid thieno probes as ligands for D2-like receptors with affinities in the subnanomolar range

enthalten in: Chemistry & biodiversity | 2013

von Abdel-Fattah, M. | Lehmann, J. | Abadi, A.

3

Chiral indolo[3,2-f][3]benzazecine-type dopamine receptor antagonists : synthesis and activity of racemic and enantiopure derivatives

enthalten in: Journal of medicinal chemistry | 2011

von Robaa, D. | Enzensperger, C. | Eldin Abulazm, S. | +4

4

Residues at the indole-NH of LE300 modulate affinities and selectivities for dopamine receptors

enthalten in: Archiv der Pharmazie | 2011

von Robaa, D. | Kretschmer, R. | Siol, O. | +4

5

Dopamine receptor ligands. Part 18 : (1) modification of the structural skeleton of indolobenzazecine-type dopamine receptor antagonists

enthalten in: Journal of medicinal chemistry | 2010

von Robaa, D. | Enzensperger, C. | Abul Azm, S. | +3

6

Arylalkylamine-, beta-carboline-, quinolizine- and azecine-derived compounds and their in vitro interaction with the ionotropic 5-HT3 receptor : search for new lead structures

enthalten in: Arzneimittel-Forschung | 2010

von Enzensperger, C. | Lehmann, J. | von Schroetter, K. | +2

7

Dopamine/serotonin receptor ligands. Part 15 : Oxygenation of the benz-indolo-azecine LE 300 leads to novel subnanomolar dopamine D1/D5 antagonists

enthalten in: Bioorganic & medicinal chemistry letters | 2007

von Enzensperger, C. | Kilian, S. | Ackermann, M. | +3

8

Dopamine/serotonin receptor ligands. 13 : Homologization of a benzindoloazecine-type dopamine receptor antagonist modulates the affinities for dopamine D(1)-D(5) receptors

enthalten in: Journal of medicinal chemistry | 2006

von Enzensperger, C. | Lehmann, J.

9

Dopamine/serotonin receptor ligands. 10 : SAR Studies on azecine-type dopamine receptor ligands by functional screening at human cloned D1, D2L, and D5 receptors with a microplate reader based calcium assay lead to a novel potent D1/D5 selective antagonist

enthalten in: Journal of medicinal chemistry | 2006

von Hoefgen, B. | Decker, M. | Mohr, P. | +7

10

Dopamine/serotonin receptor ligands. Part VIII : the dopamine receptor antagonist LE300 - modelled and X-ray structure plus further pharmacological characterization, including serotonin receptor binding, biogenic amine transporter testing and in vivo testings

enthalten in: European journal of medicinal chemistry | 2004

von Decker, M. | Schleifer, K. | Nieger, M. | +1