Suchergebnisse - "Lavecchia, Antonio"

PubPharm (217)

21

Discovery of a Novel Inhibitor of Human Purine Nucleoside Phosphorylase by a Simple Hydrophilic Interaction Liquid Chromatography Enzymatic Assay

enthalten in: ChemMedChem | 2021

von Rabuffetti, M. | Rinaldi, F. | Lo Bianco, A. | +7

22

HDAC4 Inhibitors with Cyclic Linker and Non‐hydroxamate Zinc Binding Group : Design, Synthesis, HDAC Screening and in vitro Cytotoxicity evaluation.

enthalten in: ChemistrySelect | 2021

von Tilekar, K. | Hess, J. | Upadhyay, N. | +8

23

Inhibition mechanism of naphthylphenylamine derivatives acting on the CDC25B dual phosphatase and analysis of the molecular processes involved in the high cytotoxicity exerted by one selected derivative in melanoma cells

enthalten in: Journal of enzyme inhibition and medicinal chemistry | 2020

von Aliotta, F. | Nasso, R. | Rullo, R. | +8

24

Inhibition of 37/67kDa Laminin-1 Receptor Restores APP Maturation and Reduces Amyloid-β in Human Skin Fibroblasts from Familial Alzheimer's Disease

enthalten in: Journal of personalized medicine | 2020

von Bhattacharya, A. | Izzo, A. | Mollo, N. | +11

25

Synthesis and Biological Evaluation of Pyrazoline and Pyrrolidine-2,5-dione Hybrids as Potential Antitumor Agents

enthalten in: ChemMedChem | 2020

von Tilekar, K. | Upadhyay, N. | Meyer-Almes, F. | +9

26

Sulfonimide and Amide Derivatives as Novel PPARα Antagonists : Synthesis, Antiproliferative Activity, and Docking Studies

enthalten in: ACS medicinal chemistry letters | 2020

von Ammazzalorso, A. | Bruno, I. | Florio, R. | +13

27

APP Maturation and Intracellular Localization Are Controlled by a Specific Inhibitor of 37/67 kDa Laminin-1 Receptor in Neuronal Cells

enthalten in: International journal of molecular sciences | 2020

von Bhattacharya, A. | Limone, A. | Napolitano, F. | +6

28

Antitumor agents 7. Synthesis, antiproliferative activity and molecular modeling of new l-lysine-conjugated pyridophenoxazinones as potent DNA-binding ligands and topoisomerase IIα inhibitors

enthalten in: European journal of medicinal chemistry | 2020

von Pedatella, S. | Cerchia, C. | Manfra, M. | +3

29

Synthesis and Biological Evaluation of Pyrazoline and Pyrrolidine‐2,5‐dione Hybrids as Potential Antitumor Agents

enthalten in: ChemMedChem | 2020

von Tilekar, K. | Upadhyay, N. | Meyer‐Almes, F. | +9

30

Deep learning in drug discovery : opportunities, challenges and future prospects

enthalten in: Drug discovery today | 2019

von Lavecchia, A.