Suchergebnisse - "Lavecchia, Antonio"

PubPharm (34)

1

Identification of selective 5-LOX and FLAP inhibitors as novel anti-inflammatory agents by ligand-based virtual screening

enthalten in: European journal of medicinal chemistry | 2024

von Cerchia, C. | Küfner, L. | Werz, O. | +1

2

Impairment of Nucleolin Activity and Phosphorylation by a Trachylobane Diterpene from Psiadia punctulata in Cancer Cells

enthalten in: International journal of molecular sciences | 2022

von Bellone, M. | Fiengo, L. | Cerchia, C. | +5

3

A chemoinformatics search for peroxisome proliferator-activated receptors ligands revealed a new pan-agonist able to reduce lipid accumulation and improve insulin sensitivity

enthalten in: European journal of medicinal chemistry | 2022

von Sblano, S. | Cerchia, C. | Laghezza, A. | +11

4

Antitumor agents 7. Synthesis, antiproliferative activity and molecular modeling of new l-lysine-conjugated pyridophenoxazinones as potent DNA-binding ligands and topoisomerase IIα inhibitors

enthalten in: European journal of medicinal chemistry | 2020

von Pedatella, S. | Cerchia, C. | Manfra, M. | +3

5

Selective PPARγ modulators for Type 2 diabetes treatment : how far have we come and what does the future hold?

enthalten in: Future medicinal chemistry | 2018

von Lavecchia, A. | Cerchia, C.

6

A compound-based proteomic approach discloses 15-ketoatractyligenin methyl ester as a new PPARγ partial agonist with anti-proliferative ability

enthalten in: Scientific reports | 2017

von Vasaturo, M. | Fiengo, L. | De Tommasi, N. | +9

7

Structural basis for PPAR partial or full activation revealed by a novel ligand binding mode

enthalten in: Scientific reports | 2016

von Capelli, D. | Cerchia, C. | Montanari, R. | +6

8

The antiproliferative and proapoptotic effects of cladosporols A and B are related to their different binding mode as PPARγ ligands

enthalten in: Biochemical pharmacology | 2016

von Zurlo, D. | Ziccardi, P. | Votino, C. | +9

9

In silico methods to address polypharmacology : current status, applications and future perspectives

enthalten in: Drug discovery today | 2016

von Lavecchia, A. | Cerchia, C.

10

Ligand-based chemoinformatic discovery of a novel small molecule inhibitor targeting CDC25 dual specificity phosphatases and displaying in vitro efficacy against melanoma cells

enthalten in: Oncotarget | 2015

von Capasso, A. | Cerchia, C. | Di Giovanni, C. | +6