Suchergebnisse - "Lavecchia, Antonio"

PubPharm (35)

1

Thiazolidinedione "Magic Bullets" Simultaneously Targeting PPARγ and HDACs : Design, Synthesis, and Investigations of their In Vitro and In Vivo Antitumor Effects

enthalten in: Journal of medicinal chemistry | 2021

von Tilekar, K. | Hess, J. | Upadhyay, N. | +8

2

Discovery of a Novel Inhibitor of Human Purine Nucleoside Phosphorylase by a Simple Hydrophilic Interaction Liquid Chromatography Enzymatic Assay

enthalten in: ChemMedChem | 2021

von Rabuffetti, M. | Rinaldi, F. | Lo Bianco, A. | +7

3

Pharmacophore hybridization approach to discover novel pyrazoline-based hydantoin analogs with anti-tumor efficacy

enthalten in: Bioorganic chemistry | 2021

von Upadhyay, N. | Tilekar, K. | Loiodice, F. | +9

4

Inhibition mechanism of naphthylphenylamine derivatives acting on the CDC25B dual phosphatase and analysis of the molecular processes involved in the high cytotoxicity exerted by one selected derivative in melanoma cells

enthalten in: Journal of enzyme inhibition and medicinal chemistry | 2020

von Aliotta, F. | Nasso, R. | Rullo, R. | +8

5

Synthesis and Biological Evaluation of Pyrazoline and Pyrrolidine-2,5-dione Hybrids as Potential Antitumor Agents

enthalten in: ChemMedChem | 2020

von Tilekar, K. | Upadhyay, N. | Meyer-Almes, F. | +9

6

Antitumor agents 7. Synthesis, antiproliferative activity and molecular modeling of new l-lysine-conjugated pyridophenoxazinones as potent DNA-binding ligands and topoisomerase IIα inhibitors

enthalten in: European journal of medicinal chemistry | 2020

von Pedatella, S. | Cerchia, C. | Manfra, M. | +3

7

Discovery of Novel Naphthylphenylketone and Naphthylphenylamine Derivatives as Cell Division Cycle 25B (CDC25B) Phosphatase Inhibitors : Design, Synthesis, Inhibition Mechanism, and in Vitro Efficacy against Melanoma Cell Lines

enthalten in: Journal of medicinal chemistry | 2019

von Cerchia, C. | Nasso, R. | Mori, M. | +10

8

Urokinase-type plasminogen activator receptor (uPAR) expression enhances invasion and metastasis in RAS mutated tumors

enthalten in: Scientific reports | 2017

von Mauro, C. | Pesapane, A. | Formisano, L. | +20

9

CDC25 Inhibition in Acute Myeloid Leukemia-A Study of Patient Heterogeneity and the Effects of Different Inhibitors

enthalten in: Molecules (Basel, Switzerland) | 2017

von Brenner, A. | Reikvam, H. | Rye, K. | +3

10

New diphenylmethane derivatives as peroxisome proliferator-activated receptor alpha/gamma dual agonists endowed with anti-proliferative effects and mitochondrial activity

enthalten in: European journal of medicinal chemistry | 2017

von Piemontese, L. | Cerchia, C. | Laghezza, A. | +11