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topic_facet:"Adenosine A1 Receptor Agonists"
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PubPharm (5)
1
Structure-Based Design, Synthesis, and In Vivo Antinociceptive Effects of Selective A1 Adenosine Receptor Agonists
enthalten in:
Journal of medicinal chemistry
| 2018
von
Petrelli, R.
|
Scortichini, M.
|
Belardo, C.
| +10
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2
Exploring the Role of N6-Substituents in Potent Dual Acting 5'-C-Ethyltetrazolyladenosine Derivatives : Synthesis, Binding, Functional Assays, and Antinociceptive Effects in Mice ∇
enthalten in:
Journal of medicinal chemistry
| 2017
von
Petrelli, R.
|
Scortichini, M.
|
Kachler, S.
| +12
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3
5'-C-Ethyl-tetrazolyl-N(6)-substituted adenosine and 2-chloro-adenosine derivatives as highly potent dual acting A1 adenosine receptor agonists and A3 adenosine receptor antagonists
enthalten in:
Journal of medicinal chemistry
| 2015
von
Petrelli, R.
|
Torquati, I.
|
Kachler, S.
| +8
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4
N6-Cycloalkyl- and N6-bicycloalkyl-C5'(C2')-modified adenosine derivatives as high-affinity and selective agonists at the human A1 adenosine receptor with antinociceptive effects in mice
enthalten in:
Journal of medicinal chemistry
| 2009
von
Franchetti, P.
|
Cappellacci, L.
|
Vita, P.
| +8
ErratumIn: J Med Chem. 2009 May 28;52(10):3430
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5
5'-Carbamoyl derivatives of 2'-C-methyl-purine nucleosides as selective A1 adenosine receptor agonists : affinity, efficacy, and selectivity for A1 receptor from different species
enthalten in:
Bioorganic & medicinal chemistry
| 2008
von
Cappellacci, L.
|
Franchetti, P.
|
Vita, P.
| +7
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1
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Thema: Adenosine A1 Receptor Agonists
Medienart
5
Aufsätze
5
E-Artikel
5
E-Ressourcen
Zeitschriftentitel
4
Journal of medicinal chemistry
1
Bioorganic & medicinal chemistry
Thema
Adenosine A1 Receptor Agonists
5
Journal Article
5
Research Support, Non-U.S. Gov't
4
Adenosine
4
K72T3FS567
3
Analgesics
3
Receptor, Adenosine A1
2
Adenosine A3 Receptor Antagonists
2
Adenylyl Cyclases
2
EC 4.6.1.1
2
Receptor, Adenosine A3
1
Carbamates
1
Cyclopentanes
1
Norbornanes
1
Purine Nucleosides
1
Purinergic P1 Receptor Agonists
1
Purinergic P1 Receptor Antagonists
1
Receptors, Purinergic P1
1
Research Support, N.I.H., Intramural
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Erscheinungszeitraum
3
2010-2019
2
2000-2009
Erscheinungsjahr(e)
Von:
Bis:
Sprache
5
Englisch
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