Suchergebnisse - "Knapp, Stefan"

PubPharm (780)

11

Tracking the PROTAC degradation pathway in living cells highlights the importance of ternary complex measurement for PROTAC optimization

enthalten in: bioRxiv.org | 2024

von Schwalm, M. | Krämer, A. | Dölle, A. | +5

12

Death by a Thousand Cuts – Combining Kinase Inhibitors for Selective Target Inhibition and Rational Polypharmacology

enthalten in: bioRxiv.org | 2024

von Outhwaite, I. | Singh, S. | Berger, B. | +3

13

5-iodotubercidin sensitizes cells to RIPK1-dependent necroptosis by interfering with NFκB signaling

enthalten in: bioRxiv.org | 2024

von Chauhan, C. | Kraemer, A. | Knapp, S. | +4

14

Shifting the selectivity of pyrido[2,3-d]pyrimidin-7(8H)-one inhibitors towards the salt-inducible kinase (SIK) subfamily

enthalten in: bioRxiv.org | 2024

von Rak, M. | Tesch, R. | Berger, L. | +15

15

Luciferase- and HaloTag-based reporter assays to measure small-molecule-induced degradation pathway in living cells

enthalten in: Nature protocols | 2024

von Schwalm, M. | Saxena, K. | Müller, S. | +1

16

Discovery of a Small Molecule Activator of Slack (Kcnt1) Potassium Channels That Significantly Reduces Scratching in Mouse Models of Histamine-Independent and Chronic Itch

enthalten in: Advanced science (Weinheim, Baden-Wurttemberg, Germany) | 2024

von Balzulat, A. | Zhu, W. | Flauaus, C. | +18

17

Discovery of the sEH Inhibitor Epoxykynin as a Potent Kynurenine Pathway Modulator

enthalten in: Journal of medicinal chemistry | 2024

von Dötsch, L. | Davies, C. | Hennes, E. | +12

18

tracerDB: A crowdsourced fluorescent tracer database for target engagement analysis

enthalten in: ResearchSquare.com | 2024

von Schwalm, M. | Dopfer, J. | Vasta, J. | +3

19

Development of Highly Potent and Selective FGFR4 Inhibitors Based on SNAr Electrophiles

enthalten in: chemRxiv.org | 2024

von Schwarz, M. | Kurkunov, M. | Wittlinger, F. | +9

20

Development of Highly Potent and Selective Covalent FGFR4 Inhibitors Based on SNAr Electrophiles

enthalten in: chemRxiv.org | 2024

von Schwarz, M. | Kurkunov, M. | Wittlinger, F. | +9