Suchergebnisse - "Janetka, James W"

PubPharm (15)

1

Macrocyclic Inhibitors of HGF-Activating Serine Proteases Overcome Resistance to Receptor Tyrosine Kinase Inhibitors and Block Lung Cancer Progression

enthalten in: Journal of medicinal chemistry | 2021

von Damalanka, V. | Voss, J. | Mahoney, M. | +4

2

A novel class of TMPRSS2 inhibitors potently block SARS-CoV-2 and MERS-CoV viral entry and protect human epithelial lung cells

enthalten in: Proceedings of the National Academy of Sciences of the United States of America | 2021

von Mahoney, M. | Damalanka, V. | Tartell, M. | +20

UpdateOf: bioRxiv. 2021 May 06;:. - PMID 34131661

3

A host receptor enables type 1 pilus-mediated pathogenesis of Escherichia coli pyelonephritis

enthalten in: PLoS pathogens | 2021

von McLellan, L. | McAllaster, M. | Kim, A. | +10

4

Identification of small molecule enzyme inhibitors as broad-spectrum anthelmintics

enthalten in: Scientific reports | 2019

von Tyagi, R. | Elfawal, M. | Wildman, S. | +8

5

Discovery of Selective Matriptase and Hepsin Serine Protease Inhibitors : Useful Chemical Tools for Cancer Cell Biology

enthalten in: Journal of medicinal chemistry | 2019

von Damalanka, V. | Han, Z. | Karmakar, P. | +8

6

Hepatocyte growth factor activator inhibitor-2 stabilizes Epcam and maintains epithelial organization in the mouse intestine

enthalten in: Communications biology | 2019

von Kawaguchi, M. | Yamamoto, K. | Takeda, N. | +7

7

Selective depletion of uropathogenic E. coli from the gut by a FimH antagonist

enthalten in: Nature | 2017

von Spaulding, C. | Klein, R. | Ruer, S. | +10

CommentIn: Nature. 2017 Jun 22;546(7659):479-480. - PMID 28614303

8

Photoaffinity labeling with cholesterol analogues precisely maps a cholesterol-binding site in voltage-dependent anion channel-1

enthalten in: The Journal of biological chemistry | 2017

von Budelier, M. | Cheng, W. | Bergdoll, L. | +8

9

α-Ketobenzothiazole Serine Protease Inhibitors of Aberrant HGF/c-MET and MSP/RON Kinase Pathway Signaling in Cancer

enthalten in: ChemMedChem | 2016

von Han, Z. | Harris, P. | Karmakar, P. | +5

10

Structure-based discovery of small molecule hepsin and HGFA protease inhibitors : Evaluation of potency and selectivity derived from distinct binding pockets

enthalten in: Bioorganic & medicinal chemistry | 2015

von Franco, F. | Jones, D. | Harris, P. | +4