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topic_facet:"ALDH1A1 protein, human"
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PubPharm (9)
1
Structure-Based Optimization of a Novel Class of Aldehyde Dehydrogenase 1A (ALDH1A) Subfamily-Selective Inhibitors as Potential Adjuncts to Ovarian Cancer Chemotherapy
enthalten in:
Journal of medicinal chemistry
| 2018
von
Huddle, B.
|
Grimley, E.
|
Buchman, C.
| +13
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2
Inhibition of the Aldehyde Dehydrogenase 1/2 Family by Psoralen and Coumarin Derivatives
enthalten in:
Journal of medicinal chemistry
| 2017
von
Buchman, C.
|
Hurley, T.
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3
Development of a high-throughput in vitro assay to identify selective inhibitors for human ALDH1A1
enthalten in:
Chemico-biological interactions
| 2015
von
Morgan, C.
|
Hurley, T.
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4
Discovery of a series of aromatic lactones as ALDH1/2-directed inhibitors
enthalten in:
Chemico-biological interactions
| 2015
von
Buchman, C.
|
Mahalingan, K.
|
Hurley, T.
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5
Characterization of two distinct structural classes of selective aldehyde dehydrogenase 1A1 inhibitors
enthalten in:
Journal of medicinal chemistry
| 2015
von
Morgan, C.
|
Hurley, T.
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6
Development of selective inhibitors for human aldehyde dehydrogenase 3A1 (ALDH3A1) for the enhancement of cyclophosphamide cytotoxicity
enthalten in:
Chembiochem : a European journal of chemical biology
| 2014
von
Parajuli, B.
|
Georgiadis, T.
|
Fishel, M.
| +1
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7
Discovery of a novel class of covalent inhibitor for aldehyde dehydrogenases
enthalten in:
The Journal of biological chemistry
| 2011
von
Khanna, M.
|
Chen, C.
|
Kimble-Hill, A.
| +8
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8
Selective alteration of the rate-limiting step in cytosolic aldehyde dehydrogenase through random mutagenesis
enthalten in:
Biochemistry
| 2006
von
Ho, K.
|
Hurley, T.
|
Weiner, H.
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9
Differential effects of Mg2+ ions on the individual kinetic steps of human cytosolic and mitochondrial aldehyde dehydrogenases
enthalten in:
Biochemistry
| 2005
von
Ho, K.
|
Allali-Hassani, A.
|
Hurley, T.
| +1
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1
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Thema: ALDH1A1 protein, human
Medienart
9
Aufsätze
7
E-Artikel
7
E-Ressourcen
2
Gedruckte Aufsätze
Zeitschriftentitel
3
Journal of medicinal chemistry
2
Biochemistry
2
Chemico-biological interactions
1
Chembiochem : a European journal of chemical bi...
1
The Journal of biological chemistry
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Thema
ALDH1A1 protein, human
9
Aldehyde Dehydrogenase
9
Aldehyde Dehydrogenase 1 Family
9
EC 1.2.1
9
EC 1.2.1.3
9
EC 1.2.1.36
9
Journal Article
9
Retinal Dehydrogenase
8
Research Support, N.I.H., Extramural
6
Enzyme Inhibitors
6
Isoenzymes
4
Aldehyde Dehydrogenase, Mitochondrial
4
Research Support, U.S. Gov't, Non-P.H.S.
3
0U46U6E8UK
3
ALDH2 protein, human
3
NAD
2
8N3DW7272P
2
ALDH3A1 protein, human
2
Acetaldehyde
2
Aldehyde dehydrogenase
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Erscheinungszeitraum
7
2010-2019
2
2000-2009
Erscheinungsjahr(e)
Von:
Bis:
Sprache
9
Englisch
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