Suchergebnisse - "Eleuteri, Michela"

PubPharm (12)

1

Use of ionic liquids in amidation reactions for proteolysis targeting chimera synthesis

enthalten in: Organic & biomolecular chemistry | 2024

von Eleuteri, M. | Desantis, J. | Cruciani, G. | +2

2

Design, synthesis, and biological evaluation of first-in-class indomethacin-based PROTACs degrading SARS-CoV-2 main protease and with broad-spectrum antiviral activity

enthalten in: European journal of medicinal chemistry | 2024

von Desantis, J. | Bazzacco, A. | Eleuteri, M. | +6

3

VHL-Modified PROteolysis TArgeting Chimeras (PROTACs) as a Strategy to Evade Metabolic Degradation in In Vitro Applications

enthalten in: Journal of medicinal chemistry | 2023

von Castellani, B. | Eleuteri, M. | Di Bona, S. | +3

4

BI-FUNCTIONAL COMPOUNDS AND METHODS FOR TARGETED UBIQUITINATION OF ANDROGEN RECEPTOR

enthalten in: Europäisches Patentamt | 2023

von DESANTIS JENNY | VAZ ROY JOSEPH | ELEUTERI MICHELA

5

BI-FUNCTIONAL COMPOUNDS AND METHODS FOR TARGETED UBIQUITINATION OF ANDROGEN RECEPTOR

enthalten in: Europäisches Patentamt | 2023

von DESANTIS JENNY | VAZ ROY JOSEPH | ELEUTERI MICHELA

6

BI-FUNCTIONAL COMPOUNDS AND METHODS FOR TARGETED UBIQUITINATION OF ANDROGEN RECEPTOR

enthalten in: Europäisches Patentamt | 2023

von DESANTIS JENNY | VAZ ROY JOSEPH | ELEUTERI MICHELA

7

BI-FUNCTIONAL COMPOUNDS AND METHODS FOR TARGETED UBIQUITINATION OF ANDROGEN RECEPTOR

enthalten in: Europäisches Patentamt | 2023

von DESANTIS JENNY | VAZ ROY JOSEPH | ELEUTERI MICHELA

8

BI-FUNCTIONAL COMPOUNDS AND METHODS FOR TARGETED UBIQUITINATION OF ANDROGEN RECEPTOR

enthalten in: Europäisches Patentamt | 2023

von DESANTIS JENNY | VAZ ROY JOSEPH | ELEUTERI MICHELA

9

Discovery of novel SARS-CoV-2 inhibitors targeting the main protease Mpro by virtual screenings and hit optimization

enthalten in: Antiviral research | 2022

von Mercorelli, B. | Desantis, J. | Celegato, M. | +8

10

PROTACs bearing piperazine-containing linkers : what effect on their protonation state?

enthalten in: RSC advances | 2022

von Desantis, J. | Mammoli, A. | Eleuteri, M. | +4