Suchergebnisse - "Canale, Vittorio"

PubPharm (65)

41

Synthesis and Pharmacological Evaluation of Novel Silodosin-Based Arylsulfonamide Derivatives as α1A/α1D-Adrenergic Receptor Antagonist with Potential Uroselective Profile

enthalten in: Molecules (Basel, Switzerland) | 2018

von Canale, V. | Rak, A. | Kotańska, M. | +9

42

Biotransformation of 4-fluoro-N-(1-{2-[(propan-2-yl)phenoxy]ethyl}-8-azabicyclo[3.2.1]octan-3-yl)-benzenesulfonamide, a novel potent 5-HT7 receptor antagonist with antidepressant-like and anxiolytic properties : In vitro and in silico approach

enthalten in: Journal of biochemical and molecular toxicology | 2018

von Słoczyńska, K. | Wójcik-Pszczoła, K. | Canale, V. | +3

43

Novel multi-target azinesulfonamides of cyclic amine derivatives as potential antipsychotics with pro-social and pro-cognitive effects

enthalten in: European journal of medicinal chemistry | 2018

von Zajdel, P. | Kos, T. | Marciniec, K. | +16

44

Novel non-sulfonamide 5-HT6 receptor partial inverse agonist in a group of imidazo[4,5-b]pyridines with cognition enhancing properties

enthalten in: European journal of medicinal chemistry | 2018

von Vanda, D. | Soural, M. | Canale, V. | +12

45

The impact of the halogen bonding on D2 and 5-HT1A/5-HT7 receptor activity of azinesulfonamides of 4-[(2-ethyl)piperidinyl-1-yl]phenylpiperazines with antipsychotic and antidepressant properties

enthalten in: Bioorganic & medicinal chemistry | 2017

von Partyka, A. | Kurczab, R. | Canale, V. | +8

46

Novel 5-HT7R antagonists, arylsulfonamide derivatives of (aryloxy)propyl piperidines : Add-on effect to the antidepressant activity of SSRI and DRI, and pro-cognitive profile

enthalten in: Bioorganic & medicinal chemistry | 2017

von Canale, V. | Partyka, A. | Kurczab, R. | +9

47

Arylsulfonamide derivatives of (aryloxy)ethyl pyrrolidines and piperidines as α1-adrenergic receptor antagonist with uro-selective activity

enthalten in: Bioorganic & medicinal chemistry | 2016

von Rak, A. | Canale, V. | Marciniec, K. | +10

48

N1-Azinylsulfonyl-1H-indoles : 5-HT6 Receptor Antagonists with Procognitive and Antidepressant-Like Properties

enthalten in: ACS medicinal chemistry letters | 2016

von Zajdel, P. | Marciniec, K. | Satała, G. | +10

49

Preliminary mutagenicity and genotoxicity evaluation of selected arylsulfonamide derivatives of (aryloxy)alkylamines with potential psychotropic properties

enthalten in: Journal of applied genetics | 2016

von Powroźnik, B. | Słoczyńska, K. | Canale, V. | +3

50

Towards new 5-HT7 antagonists among arylsulfonamide derivatives of (aryloxy)ethyl-alkyl amines : Multiobjective based design, synthesis, and antidepressant and anxiolytic properties

enthalten in: European journal of medicinal chemistry | 2016

von Canale, V. | Kurczab, R. | Partyka, A. | +6