Suchergebnisse - "Canale, Vittorio"

PubPharm (18)

1

The Constitutive Activity of Spinal 5-HT6 Receptors Contributes to Diabetic Neuropathic Pain in Rats

enthalten in: Biomolecules | 2023

von Mokhtar, N. | Drop, M. | Jacquot, F. | +10

2

1-(Arylsulfonyl-isoindol-2-yl)piperazines as 5-HT6R Antagonists : Mechanochemical Synthesis, In Vitro Pharmacological Properties and Glioprotective Activity

enthalten in: Biomolecules | 2022

von Canale, V. | Trybała, W. | Chaumont-Dubel, S. | +10

3

Neuropathic pain-alleviating activity of novel 5-HT6 receptor inverse agonists derived from 2-aryl-1H-pyrrole-3-carboxamide

enthalten in: Bioorganic chemistry | 2021

von Drop, M. | Jacquot, F. | Canale, V. | +20

4

2-Phenyl-1H-pyrrole-3-carboxamide as a New Scaffold for Developing 5-HT6 Receptor Inverse Agonists with Cognition-Enhancing Activity

enthalten in: ACS chemical neuroscience | 2021

von Drop, M. | Canale, V. | Chaumont-Dubel, S. | +19

5

Imidazopyridine-Based 5-HT6 Receptor Neutral Antagonists : Impact of N1-Benzyl and N1-Phenylsulfonyl Fragments on Different Receptor Conformational States

enthalten in: Journal of medicinal chemistry | 2021

von Vanda, D. | Canale, V. | Chaumont-Dubel, S. | +12

6

mTOR activation by constitutively active serotonin6 receptors as new paradigm in neuropathic pain and its treatment

enthalten in: Progress in neurobiology | 2020

von Martin, P. | Doly, S. | Hamieh, A. | +11

7

Sustainable Synthesis of a Potent and Selective 5-HT7 Receptor Antagonist Using a Mechanochemical Approach

enthalten in: The Journal of organic chemistry | 2020

von Canale, V. | Frisi, V. | Bantreil, X. | +2

8

Novel antagonists of 5-HT6 and/or 5-HT7 receptors affect the brain monoamines metabolism and enhance the anti-immobility activity of different antidepressants in rats

enthalten in: Behavioural brain research | 2019

von Partyka, A. | Jastrzębska-Więsek, M. | Antkiewicz-Michaluk, L. | +6

9

Amino Acid Hot Spots of Halogen Bonding : A Combined Theoretical and Experimental Case Study of the 5-HT7 Receptor

enthalten in: Journal of medicinal chemistry | 2018

von Kurczab, R. | Canale, V. | Satała, G. | +2

10

The impact of the halogen bonding on D2 and 5-HT1A/5-HT7 receptor activity of azinesulfonamides of 4-[(2-ethyl)piperidinyl-1-yl]phenylpiperazines with antipsychotic and antidepressant properties

enthalten in: Bioorganic & medicinal chemistry | 2017

von Partyka, A. | Kurczab, R. | Canale, V. | +8