Suchergebnisse - "Bouzriba, Chahrazed"

PubPharm (13)

1

Design, synthesis and biological evaluation of new 2,6-difluorinated phenyl 4-(2-oxoimidazolidin-1-yl)benzenesulfonates as new antimicrotubule agents

enthalten in: Bioorganic chemistry | 2024

von Bouzriba, C. | Gagné-Boulet, M. | Chavez Alvarez, A. | +3

2

Modification of the phenyl ring B of phenyl 4-(2-oxoimidazolidin-1-yl)benzenesulfonates by pyridinyl moiety leads to novel antimitotics targeting the colchicine-binding site

enthalten in: Bioorganic & medicinal chemistry letters | 2024

von Ouellette, V. | Bouzriba, C. | Chavez Alvarez, A. | +2

3

Development of an UHPLC-UV Method for Quantification of Three Phenyl 4-(2-oxo-3-alkylimidazolidin-1-yl)benzenesulfonates in CD-$ 1^{®} $ IGS Female Mouse Plasma

enthalten in: Journal of analytical chemistry | 2024

von Alvarez, A. | Bouzriba, C. | Bernier, L. | +6

4

4-(3-Alkyl-2-oxoimidazolidin-1-yl)-N-phenylbenzenesulfonamide salts : Novel hydrosoluble prodrugs of antimitotics selectively bioactivated by the cytochrome P450 1A1 in breast cancer cells

enthalten in: Bioorganic chemistry | 2023

von Ouellette, V. | Chavez Alvarez, A. | Bouzriba, C. | +2

5

Homologation of the Alkyl Side Chain of Antimitotic Phenyl 4-(2-Oxo-3-alkylimidazolidin-1-yl)benzenesulfonate Prodrugs Selectively Targeting CYP1A1-Expressing Breast Cancers Improves Their Stability in Rodent Liver Microsomes

enthalten in: Journal of medicinal chemistry | 2023

von Chavez Alvarez, A. | Bouzriba, C. | Moreau, E. | +11

6

Preparation and biological evaluation of new antimicrotubule agents : Modification of the imidazolidin-2-one moiety of phenyl 4-(2-oxoimidazolidin-1-yl)benzenesulfonates

enthalten in: Chemical biology & drug design | 2022

von Gagné-Boulet, M. | Bouzriba, C. | Chavez Alvarez, A. | +1

7

Branched alkyl of phenyl 4-(2-oxo-3-alkylimidazolidin-1-yl)benzenesulfonates as unique cytochrome P450 1A1-activated antimitotic prodrugs : Biological evaluation and mechanism of bioactivation

enthalten in: European journal of medicinal chemistry | 2022

von Bouzriba, C. | Chavez Alvarez, A. | Gagné-Boulet, M. | +5

8

Preparation and biological evaluation of new antimicrotubule agents : Modification of the imidazolidin‐2‐one moiety of phenyl 4‐(2‐oxoimidazolidin‐1‐yl)benzenesulfonates

enthalten in: Chemical Biology & Drug Design | 2022

von Gagné‐Boulet, M. | Bouzriba, C. | Chavez Alvarez, A. | +1

9

Phenyl 4-(2-oxopyrrolidin-1-yl)benzenesulfonates and phenyl 4-(2-oxopyrrolidin-1-yl)benzenesulfonamides as new antimicrotubule agents targeting the colchicine-binding site

enthalten in: European journal of medicinal chemistry | 2021

von Gagné-Boulet, M. | Bouzriba, C. | Chavez Alvarez, A. | +1

10

N-phenyl ureidobenzenesulfonates, a novel class of promising human dihydroorotate dehydrogenase inhibitors

enthalten in: Bioorganic & medicinal chemistry | 2020

von Bouzriba, C. | Larcher, L. | Gagné-Boulet, M. | +1