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/vufind/Search/Results?lookfor=%22Blake%2C+Robert+A%22&type=Person&sort=year
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PubPharm (35)
1
Targeted degradation via direct 26S proteasome recruitment
enthalten in:
Nature chemical biology
| 2023
von
Bashore, C.
|
Prakash, S.
|
Johnson, M.
| +22
CommentIn: Nat Chem Biol. 2023 Jan;19(1):3-4. - PMID 36577874
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2
Discovery of GNE-502 as an orally bioavailable and potent degrader for estrogen receptor positive breast cancer
enthalten in:
Bioorganic & medicinal chemistry letters
| 2021
von
Zbieg, J.
|
Liang, J.
|
Li, J.
| +29
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3
GDC-9545 (Giredestrant) : A Potent and Orally Bioavailable Selective Estrogen Receptor Antagonist and Degrader with an Exceptional Preclinical Profile for ER+ Breast Cancer
enthalten in:
Journal of medicinal chemistry
| 2021
von
Liang, J.
|
Zbieg, J.
|
Blake, R.
| +44
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4
Antibody-Mediated Delivery of Chimeric BRD4 Degraders. Part 1 : Exploration of Antibody Linker, Payload Loading, and Payload Molecular Properties
enthalten in:
Journal of medicinal chemistry
| 2021
von
Dragovich, P.
|
Pillow, T.
|
Blake, R.
| +34
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5
Antibody-Mediated Delivery of Chimeric BRD4 Degraders. Part 2 : Improvement of In Vitro Antiproliferation Activity and In Vivo Antitumor Efficacy
enthalten in:
Journal of medicinal chemistry
| 2021
von
Dragovich, P.
|
Pillow, T.
|
Blake, R.
| +34
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6
Monomeric Targeted Protein Degraders
enthalten in:
Journal of medicinal chemistry
| 2020
von
Hanan, E.
|
Liang, J.
|
Wang, X.
| +3
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7
Antibody-mediated delivery of chimeric protein degraders which target estrogen receptor alpha (ERα)
enthalten in:
Bioorganic & medicinal chemistry letters
| 2020
von
Dragovich, P.
|
Adhikari, P.
|
Blake, R.
| +40
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8
Chaperone mediated detection of small molecule target binding in cells
enthalten in:
Nature communications
| 2020
von
Cho, K.
|
Ma, T.
|
Rose, C.
| +3
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9
Antibody Conjugation of a Chimeric BET Degrader Enables in vivo Activity
enthalten in:
ChemMedChem
| 2020
von
Pillow, T.
|
Adhikari, P.
|
Blake, R.
| +29
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10
Discovery of a C-8 hydroxychromene as a potent degrader of estrogen receptor alpha with improved rat oral exposure over GDC-0927
enthalten in:
Bioorganic & medicinal chemistry letters
| 2019
von
Labadie, S.
|
Li, J.
|
Blake, R.
| +19
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Bioorganic & medicinal chemistry letters
5
Journal of medicinal chemistry
4
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3
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2
eLife
1
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Cell
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Chemistry (Weinheim an der Bergstrasse, Germany)
1
Clinical cancer research : an official journal ...
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Methods in molecular biology (Clifton, N.J.)
1
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1
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1
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1
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Thema
25
Journal Article
8
Research Support, Non-U.S. Gov't
7
Antineoplastic Agents
7
Enzyme Inhibitors
6
EC 2.3.2.27
6
EC 2.7.10.1
5
Antibodies, Monoclonal
5
Estrogen Receptor alpha
5
Immunoconjugates
5
Indoles
5
Research Support, N.I.H., Extramural
5
Research Support, U.S. Gov't, Non-P.H.S.
4
Cell Cycle Proteins
4
EC 2.7.11.1
4
Transcription Factors
3
BRD4 protein, human
3
EC 6.3.2.-
3
Estrogen receptor
3
Indazoles
3
Pyrroles
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Erscheinungszeitraum
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2000-
2
1900-1999
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