Suchergebnisse - "Blaazer, Antoni R"

PubPharm (14)

1

Alkynamide phthalazinones as a new class of TbrPDEB1 inhibitors (Part 2)

enthalten in: Bioorganic & medicinal chemistry | 2019

von de Heuvel, E. | Singh, A. | Boronat, P. | +14

2

Screening of a PDE-focused library identifies imidazoles with in vitro and in vivo antischistosomal activity

enthalten in: International journal for parasitology. Drugs and drug resistance | 2019

von Botros, S. | William, S. | Sabra, A. | +17

3

Targeting a Subpocket in Trypanosoma brucei Phosphodiesterase B1 (TbrPDEB1) Enables the Structure-Based Discovery of Selective Inhibitors with Trypanocidal Activity

enthalten in: Journal of medicinal chemistry | 2018

von Blaazer, A. | Singh, A. | de Heuvel, E. | +24

4

Surface plasmon resonance biosensor assay for the analysis of small-molecule inhibitor binding to human and parasitic phosphodiesterases

enthalten in: Analytical biochemistry | 2016

von Siderius, M. | Shanmugham, A. | England, P. | +5

5

Surface plasmon resonance biosensor assay for the analysis of small-molecule inhibitor binding to human and parasitic phosphodiesterases

enthalten in: Analytical biochemistry | 2016

von Siderius, M. | Shanmugham, A. | England, P. | +5

6

Exploration of the molecular architecture of the orthosteric binding site in the α4β2 nicotinic acetylcholine receptor with analogs of 3-(dimethylamino)butyl dimethylcarbamate (DMABC) and 1-(pyridin-3-yl)-1,4-diazepane

enthalten in: European journal of medicinal chemistry | 2015

von Bach, T. | Jensen, A. | Petersen, J. | +7

7

Fragment-based screening in tandem with phenotypic screening provides novel antiparasitic hits

enthalten in: Journal of biomolecular screening | 2015

von Blaazer, A. | Orrling, K. | Shanmugham, A. | +9

8

Fragment-Based Screening in Tandem with Phenotypic Screening Provides Novel Antiparasitic Hits

enthalten in: Journal of biomolecular screening | 2015

von Blaazer, A. | Orrling, K. | Shanmugham, A. | +9

9

Exploration of the molecular architecture of the orthosteric binding site in the α4β2 nicotinic acetylcholine receptor with analogs of 3-(dimethylamino)butyl dimethylcarbamate (DMABC) and 1-(pyridin-3-yl)-1,4-diazepane

enthalten in: European journal of medicinal chemistry | 2015

von Bach, T. | Jensen, A. | Petersen, J. | +7

10

ChemInform Abstract: Novel Indole and Azaindole (Pyrrolopyridine) Cannabinoid (CB) Receptor Agonists: Design, Synthesis, Structure—Activity Relationships, Physicochemical Properties and Biological Activity.

enthalten in: ChemInform | 2012

von Blaazer, A. | Lange, J. | van der Neut, M. | +5