Suchergebnisse - "4-(3-(benzyloxy)phenyl)-2-(ethylsulfinyl)-6-(trifluoromethyl)pyrimidine"

PubPharm (8)

1

Discovery of small molecule positive allosteric modulators of the secretin receptor

enthalten in: Biochemical pharmacology | 2021

von Dengler, D. | Harikumar, K. | Pollari, S. | +6

2

Discovery and pharmacology of the covalent GLP-1 receptor (GLP-1R) allosteric modulator BETP : A novel tool to probe GLP-1R pharmacology

enthalten in: Advances in pharmacology (San Diego, Calif.) | 2020

von Willard, F. | Ho, J. | Sloop, K.

3

Positive Allosteric Modulation of the Glucagon-like Peptide-1 Receptor by Diverse Electrophiles

enthalten in: The Journal of biological chemistry | 2016

von Bueno, A. | Showalter, A. | Wainscott, D. | +6

4

Allosteric Optical Control of a Class B G-Protein-Coupled Receptor

enthalten in: Angewandte Chemie (International ed. in English) | 2016

von Broichhagen, J. | Johnston, N. | von Ohlen, Y. | +6

5

A potentiator of orthosteric ligand activity at GLP-1R acts via covalent modification

enthalten in: Nature chemical biology | 2014

von Nolte, W. | Fortin, J. | Stevens, B. | +8

CommentIn: Nat Chem Biol. 2014 Aug;10(8):609-10. - PMID 25036308

6

Allostery : A GPCR's back door

enthalten in: Nature chemical biology | 2014

von Mohr, K. | Kostenis, E.

CommentOn: Nat Chem Biol. 2014 Aug;10(8):629-31. - PMID 24997604

7

Demonstration of the innate electrophilicity of 4-(3-(benzyloxy)phenyl)-2-(ethylsulfinyl)-6-(trifluoromethyl)pyrimidine (BETP), a small-molecule positive allosteric modulator of the glucagon-like peptide-1 receptor

enthalten in: Drug metabolism and disposition: the biological fate of chemicals | 2013

von Eng, H. | Sharma, R. | McDonald, T. | +10

8

Two small molecule agonists of glucagon-like peptide-1 receptor modulate the receptor activation response differently

enthalten in: Biochemical and biophysical research communications | 2012

von Cheong, Y. | Kim, M. | Son, M. | +1

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