Suchergebnisse - (Person:"Spalluto, Giampiero")

PubPharm (24)

1

Developing novel classes of protein kinase CK1δ inhibitors by fusing [1,2,4]triazole with different bicyclic heteroaromatic systems

enthalten in: European journal of medicinal chemistry | 2021

von Grieco, I. | Bissaro, M. | Tiz, D. | +11

2

Targeting G Protein-Coupled Receptors with Magnetic Carbon Nanotubes : The Case of the A3 Adenosine Receptor

enthalten in: ChemMedChem | 2020

von Pineux, F. | Federico, S. | Klotz, K. | +7

3

1,2,4]Triazolo[1,5-c]pyrimidines as adenosine receptor antagonists : Modifications at the 8 position to reach selectivity towards A3 adenosine receptor subtype

enthalten in: European journal of medicinal chemistry | 2018

von Federico, S. | Margiotta, E. | Salmaso, V. | +5

4

5,7-Disubstituted-[1,2,4]triazolo[1,5-a][1,3,5]triazines as pharmacological tools to explore the antagonist selectivity profiles toward adenosine receptors

enthalten in: European journal of medicinal chemistry | 2016

von Federico, S. | Ciancetta, A. | Porta, N. | +6

5

Scaffold decoration at positions 5 and 8 of 1,2,4-triazolo[1,5-c]pyrimidines to explore the antagonist profiling on adenosine receptors : a preliminary structure-activity relationship study

enthalten in: Journal of medicinal chemistry | 2014

von Federico, S. | Ciancetta, A. | Porta, N. | +6

6

Revisiting a receptor-based pharmacophore hypothesis for human A(2A) adenosine receptor antagonists

enthalten in: Journal of chemical information and modeling | 2013

von Bacilieri, M. | Ciancetta, A. | Paoletta, S. | +9

7

Novel fluorescent antagonist as a molecular probe in A(3) adenosine receptor binding assays using flow cytometry

enthalten in: Biochemical pharmacology | 2012

von Kozma, E. | Kumar, T. | Federico, S. | +7

8

Does the combination of optimal substitutions at the C²-, N⁵- and N⁸-positions of the pyrazolo-triazolo-pyrimidine scaffold guarantee selective modulation of the human A₃ adenosine receptors?

enthalten in: Bioorganic & medicinal chemistry | 2011

von Cheong, S. | Dolzhenko, A. | Paoletta, S. | +8

9

Pharmacophore elucidation for a new series of 2-aryl-pyrazolo-triazolo-pyrimidines as potent human A3 adenosine receptor antagonists

enthalten in: Bioorganic & medicinal chemistry letters | 2011

von Cheong, S. | Federico, S. | Venkatesan, G. | +5

10

Synthesis and biological evaluation of a new series of 1,2,4-triazolo[1,5-a]-1,3,5-triazines as human A(2A) adenosine receptor antagonists with improved water solubility

enthalten in: Journal of medicinal chemistry | 2011

von Federico, S. | Paoletta, S. | Cheong, S. | +9