Suchergebnisse - (Person:"Maga, Giovanni")

PubPharm (20)

1

Synthesis and biological activity evaluation of 3-(hetero) arylideneindolin-2-ones as potential c-Src inhibitors

enthalten in: Journal of enzyme inhibition and medicinal chemistry | 2022

von Princiotto, S. | Musso, L. | Manetti, F. | +7

ErratumIn: J Enzyme Inhib Med Chem. 2022 Dec;37(1):2793-2794. - PMID 36229993

2

Novel pyrazolo[3,4-d]pyrimidines as dual Src/Bcr-Abl kinase inhibitors : Synthesis and biological evaluation for chronic myeloid leukemia treatment

enthalten in: Bioorganic chemistry | 2022

von Di Maria, S. | Picarazzi, F. | Mori, M. | +15

3

Identification of a new family of pyrazolo[3,4-d]pyrimidine derivatives as multitarget Fyn-Blk-Lyn inhibitors active on B- and T-lymphoma cell lines

enthalten in: European journal of medicinal chemistry | 2019

von Fallacara, A. | Passannanti, R. | Mori, M. | +12

4

Efficient optimization of pyrazolo[3,4-d]pyrimidines derivatives as c-Src kinase inhibitors in neuroblastoma treatment

enthalten in: Bioorganic & medicinal chemistry letters | 2018

von Molinari, A. | Fallacara, A. | Di Maria, S. | +10

5

Identification of new pyrrolo[2,3-d]pyrimidines as Src tyrosine kinase inhibitors in vitro active against Glioblastoma

enthalten in: European journal of medicinal chemistry | 2017

von Musumeci, F. | Fallacara, A. | Brullo, C. | +8

6

Novel pyrazolo[3,4-d]pyrimidines as dual Src-Abl inhibitors active against mutant form of Abl and the leukemia K-562 cell line

enthalten in: European journal of medicinal chemistry | 2016

von El-Moghazy, S. | George, R. | Osman, E. | +5

7

The human tyrosine kinase Kit and its gatekeeper mutant T670I, show different kinetic properties : Implications for drug design

enthalten in: Bioorganic & medicinal chemistry | 2016

von Kissova, M. | Maga, G. | Crespan, E.

8

Studies on the ATP Binding Site of Fyn Kinase for the Identification of New Inhibitors and Their Evaluation as Potential Agents against Tauopathies and Tumors

enthalten in: Journal of medicinal chemistry | 2015

von Tintori, C. | La Sala, G. | Vignaroli, G. | +22

9

Combining X-ray crystallography and molecular modeling toward the optimization of pyrazolo[3,4-d]pyrimidines as potent c-Src inhibitors active in vivo against neuroblastoma

enthalten in: Journal of medicinal chemistry | 2015

von Tintori, C. | Fallacara, A. | Radi, M. | +14

10

Exploring the chemical space around the privileged pyrazolo[3,4-d]pyrimidine scaffold : toward novel allosteric inhibitors of T315I-mutated Abl

enthalten in: ACS combinatorial science | 2014

von Vignaroli, G. | Mencarelli, M. | Sementa, D. | +6