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topic_facet:"Receptor, Adenosine A3"
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PubPharm (14)
11
Does the combination of optimal substitutions at the C²-, N⁵- and N⁸-positions of the pyrazolo-triazolo-pyrimidine scaffold guarantee selective modulation of the human A₃ adenosine receptors?
enthalten in:
Bioorganic & medicinal chemistry
| 2011
von
Cheong, S.
|
Dolzhenko, A.
|
Paoletta, S.
| +8
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12
Receptor-driven identification of novel human A₃ adenosine receptor antagonists as potential therapeutic agents
enthalten in:
Methods in enzymology
| 2010
von
Paoletta, S.
|
Federico, S.
|
Spalluto, G.
| +1
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13
Combining selectivity and affinity predictions using an integrated Support Vector Machine (SVM) approach : An alternative tool to discriminate between the human adenosine A(2A) and A(3) receptor pyrazolo-triazolo-pyrimidine antagonists binding sites
enthalten in:
Bioorganic & medicinal chemistry
| 2009
von
Michielan, L.
|
Bolcato, C.
|
Federico, S.
| +9
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14
Human A3 adenosine receptor as versatile G protein-coupled receptor example to validate the receptor homology modeling technology
enthalten in:
Current pharmaceutical design
| 2009
von
Morizzo, E.
|
Federico, S.
|
Spalluto, G.
| +1
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Thema: Receptor, Adenosine A3
Medienart
14
Aufsätze
14
E-Artikel
14
E-Ressourcen
Zeitschriftentitel
2
Bioorganic & medicinal chemistry
2
ChemMedChem
2
European journal of medicinal chemistry
2
Journal of medicinal chemistry
1
Biochemical pharmacology
1
Current pharmaceutical design
1
Expert opinion on therapeutic patents
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Medicinal research reviews
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Methods in enzymology
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Molecules (Basel, Switzerland)
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Thema
14
Journal Article
Receptor, Adenosine A3
8
Research Support, Non-U.S. Gov't
6
Pyrimidines
6
Triazoles
5
Purinergic P1 Receptor Antagonists
4
Adenosine A3 Receptor Antagonists
4
Pyrazoles
4
Receptor, Adenosine A2A
3
Adenosine A2 Receptor Antagonists
3
Ligands
3
Review
2
ADORA3 protein, human
2
G protein-coupled receptor
2
Molecular modeling
2
Pyridines
2
Receptors, Adenosine A2
2
[1,2,4]triazolo[1,5-c]pyrimidine
1
1,2,4-triazolo(1,5-c)pyrimidine
1
1RTM4PAL0V
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Erscheinungszeitraum
3
2020-
9
2010-2019
2
2000-2009
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14
Englisch
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