Suchergebnisse - (Person:"Spalluto, Giampiero")

PubPharm (18)

1

Targeting G Protein-Coupled Receptors with Magnetic Carbon Nanotubes : The Case of the A3 Adenosine Receptor

enthalten in: ChemMedChem | 2020

von Pineux, F. | Federico, S. | Klotz, K. | +7

2

Scaffold decoration at positions 5 and 8 of 1,2,4-triazolo[1,5-c]pyrimidines to explore the antagonist profiling on adenosine receptors : a preliminary structure-activity relationship study

enthalten in: Journal of medicinal chemistry | 2014

von Federico, S. | Ciancetta, A. | Porta, N. | +6

3

Exploring the directionality of 5-substitutions in a new series of 5-alkylaminopyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine as a strategy to design novel human a(3) adenosine receptor antagonists

enthalten in: Journal of medicinal chemistry | 2012

von Federico, S. | Ciancetta, A. | Sabbadin, D. | +6

4

Novel fluorescent antagonist as a molecular probe in A(3) adenosine receptor binding assays using flow cytometry

enthalten in: Biochemical pharmacology | 2012

von Kozma, E. | Kumar, T. | Federico, S. | +7

5

Does the combination of optimal substitutions at the C²-, N⁵- and N⁸-positions of the pyrazolo-triazolo-pyrimidine scaffold guarantee selective modulation of the human A₃ adenosine receptors?

enthalten in: Bioorganic & medicinal chemistry | 2011

von Cheong, S. | Dolzhenko, A. | Paoletta, S. | +8

6

Receptor-driven identification of novel human A₃ adenosine receptor antagonists as potential therapeutic agents

enthalten in: Methods in enzymology | 2010

von Paoletta, S. | Federico, S. | Spalluto, G. | +1

7

Combining selectivity and affinity predictions using an integrated Support Vector Machine (SVM) approach : An alternative tool to discriminate between the human adenosine A(2A) and A(3) receptor pyrazolo-triazolo-pyrimidine antagonists binding sites

enthalten in: Bioorganic & medicinal chemistry | 2009

von Michielan, L. | Bolcato, C. | Federico, S. | +9

8

Human A3 adenosine receptor as versatile G protein-coupled receptor example to validate the receptor homology modeling technology

enthalten in: Current pharmaceutical design | 2009

von Morizzo, E. | Federico, S. | Spalluto, G. | +1

9

The application of a 3D-QSAR (autoMEP/PLS) approach as an efficient pharmacodynamic-driven filtering method for small-sized virtual library : application to a lead optimization of a human A3 adenosine receptor antagonist

enthalten in: Bioorganic & medicinal chemistry | 2006

von Moro, S. | Bacilieri, M. | Cacciari, B. | +5

10

A3 adenosine receptor antagonists delay irreversible synaptic failure caused by oxygen and glucose deprivation in the rat CA1 hippocampus in vitro

enthalten in: British journal of pharmacology | 2006

von Pugliese, A. | Coppi, E. | Spalluto, G. | +2