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topic_facet:"Receptor, Adenosine A3"
topic_facet:"Journal Article"
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PubPharm (24)
1
1,2,4]Triazolo[1,5-c]pyrimidines as Tools to Investigate A3 Adenosine Receptors in Cancer Cell Lines
enthalten in:
ChemMedChem
| 2023
von
Federico, S.
|
Persico, M.
|
Trevisan, L.
| +11
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2
Targeting G Protein-Coupled Receptors with Magnetic Carbon Nanotubes : The Case of the A3 Adenosine Receptor
enthalten in:
ChemMedChem
| 2020
von
Pineux, F.
|
Federico, S.
|
Klotz, K.
| +7
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3
Conjugable A3 adenosine receptor antagonists for the development of functionalized ligands and their use in fluorescent probes
enthalten in:
European journal of medicinal chemistry
| 2020
von
Federico, S.
|
Margiotta, E.
|
Moro, S.
| +4
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4
Design, Synthesis and Evaluation of New Indolylpyrimidylpiperazines for Gastrointestinal Cancer Therapy
enthalten in:
Molecules (Basel, Switzerland)
| 2019
von
Tan, A.
|
Babak, M.
|
Venkatesan, G.
| +10
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5
1,2,4]Triazolo[1,5-c]pyrimidines as adenosine receptor antagonists : Modifications at the 8 position to reach selectivity towards A3 adenosine receptor subtype
enthalten in:
European journal of medicinal chemistry
| 2018
von
Federico, S.
|
Margiotta, E.
|
Salmaso, V.
| +5
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6
Scaffold decoration at positions 5 and 8 of 1,2,4-triazolo[1,5-c]pyrimidines to explore the antagonist profiling on adenosine receptors : a preliminary structure-activity relationship study
enthalten in:
Journal of medicinal chemistry
| 2014
von
Federico, S.
|
Ciancetta, A.
|
Porta, N.
| +6
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7
The A3 adenosine receptor as multifaceted therapeutic target : pharmacology, medicinal chemistry, and in silico approaches
enthalten in:
Medicinal research reviews
| 2013
von
Cheong, S.
|
Federico, S.
|
Venkatesan, G.
| +5
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8
Exploring the directionality of 5-substitutions in a new series of 5-alkylaminopyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine as a strategy to design novel human a(3) adenosine receptor antagonists
enthalten in:
Journal of medicinal chemistry
| 2012
von
Federico, S.
|
Ciancetta, A.
|
Sabbadin, D.
| +6
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9
Novel fluorescent antagonist as a molecular probe in A(3) adenosine receptor binding assays using flow cytometry
enthalten in:
Biochemical pharmacology
| 2012
von
Kozma, E.
|
Kumar, T.
|
Federico, S.
| +7
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10
Therapeutic potential of A2 and A3 adenosine receptor : a review of novel patented ligands
enthalten in:
Expert opinion on therapeutic patents
| 2012
von
Federico, S.
|
Spalluto, G.
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1
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Thema: Receptor, Adenosine A3
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Thema
Journal Article
Receptor, Adenosine A3
18
Research Support, Non-U.S. Gov't
13
Pyrimidines
12
Triazoles
10
Adenosine A3 Receptor Antagonists
8
Purinergic P1 Receptor Antagonists
7
Ligands
6
Pyrazoles
5
Review
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Receptor, Adenosine A2A
4
Receptors, Purinergic P1
3
9009-81-8
3
Adenosine A2 Receptor Antagonists
3
Pyridines
3
Rhodopsin
2
ADORA3 protein, human
2
Cyclic AMP
2
E0399OZS9N
2
G protein-coupled receptor
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2020-
9
2010-2019
12
2000-2009
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24
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