Suchergebnisse - (Person:"Spalluto, Giampiero")

PubPharm (14)

1

Developing novel classes of protein kinase CK1δ inhibitors by fusing [1,2,4]triazole with different bicyclic heteroaromatic systems

enthalten in: European journal of medicinal chemistry | 2021

von Grieco, I. | Bissaro, M. | Tiz, D. | +11

2

Targeting G Protein-Coupled Receptors with Magnetic Carbon Nanotubes : The Case of the A3 Adenosine Receptor

enthalten in: ChemMedChem | 2020

von Pineux, F. | Federico, S. | Klotz, K. | +7

3

1,2,4]Triazolo[1,5-c]pyrimidines as adenosine receptor antagonists : Modifications at the 8 position to reach selectivity towards A3 adenosine receptor subtype

enthalten in: European journal of medicinal chemistry | 2018

von Federico, S. | Margiotta, E. | Salmaso, V. | +5

4

Scaffold decoration at positions 5 and 8 of 1,2,4-triazolo[1,5-c]pyrimidines to explore the antagonist profiling on adenosine receptors : a preliminary structure-activity relationship study

enthalten in: Journal of medicinal chemistry | 2014

von Federico, S. | Ciancetta, A. | Porta, N. | +6

5

Pharmacophore elucidation for a new series of 2-aryl-pyrazolo-triazolo-pyrimidines as potent human A3 adenosine receptor antagonists

enthalten in: Bioorganic & medicinal chemistry letters | 2011

von Cheong, S. | Federico, S. | Venkatesan, G. | +5

6

The significance of 2-furyl ring substitution with a 2-(para-substituted) aryl group in a new series of pyrazolo-triazolo-pyrimidines as potent and highly selective hA(3) adenosine receptors antagonists : new insights into structure-affinity relationship and receptor-antagonist recognition

enthalten in: Journal of medicinal chemistry | 2010

von Cheong, S. | Dolzhenko, A. | Kachler, S. | +8

7

Combining selectivity and affinity predictions using an integrated Support Vector Machine (SVM) approach : An alternative tool to discriminate between the human adenosine A(2A) and A(3) receptor pyrazolo-triazolo-pyrimidine antagonists binding sites

enthalten in: Bioorganic & medicinal chemistry | 2009

von Michielan, L. | Bolcato, C. | Federico, S. | +9

8

Linear and nonlinear 3D-QSAR approaches in tandem with ligand-based homology modeling as a computational strategy to depict the pyrazolo-triazolo-pyrimidine antagonists binding site of the human adenosine A2A receptor

enthalten in: Journal of chemical information and modeling | 2008

von Michielan, L. | Bacilieri, M. | Schiesaro, A. | +7

9

Synthesis and biological studies of a new series of 5-heteroarylcarbamoylaminopyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidines as human A3 adenosine receptor antagonists. Influence of the heteroaryl substituent on binding affinity and molecular modeling investigations

enthalten in: Journal of medicinal chemistry | 2006

von Pastorin, G. | Da Ros, T. | Bolcato, C. | +7

10

Ligand-based homology modeling as attractive tool to inspect GPCR structural plasticity

enthalten in: Current pharmaceutical design | 2006

von Moro, S. | Deflorian, F. | Bacilieri, M. | +1