Suchergebnisse - (Person:"Spalluto, Giampiero")

PubPharm (13)

1

Pyrazolo-triazolo-pyrimidine Scaffold as a Molecular Passepartout for the Pan-Recognition of Human Adenosine Receptors

enthalten in: Biomolecules | 2023

von Salmaso, V. | Persico, M. | Da Ros, T. | +5

2

1,2,4]Triazolo[1,5-c]pyrimidines as Tools to Investigate A3 Adenosine Receptors in Cancer Cell Lines

enthalten in: ChemMedChem | 2023

von Federico, S. | Persico, M. | Trevisan, L. | +11

3

1,2,4]Triazolo[1,5-c]pyrimidines as adenosine receptor antagonists : Modifications at the 8 position to reach selectivity towards A3 adenosine receptor subtype

enthalten in: European journal of medicinal chemistry | 2018

von Federico, S. | Margiotta, E. | Salmaso, V. | +5

4

Pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidines and Structurally Simplified Analogs. Chemistry and SAR Profile as Adenosine Receptor Antagonists

enthalten in: Current topics in medicinal chemistry | 2016

von Redenti, S. | Ciancetta, A. | Pastorin, G. | +4

5

The Influence of the 1-(3-Trifluoromethyl-Benzyl)-1H-Pyrazole-4-yl Moiety on the Adenosine Receptors Affinity Profile of Pyrazolo[4,3-e][1,2,4]Triazolo[1,5-c]Pyrimidine Derivatives

enthalten in: PloS one | 2015

von Federico, S. | Redenti, S. | Sturlese, M. | +6

6

Scaffold decoration at positions 5 and 8 of 1,2,4-triazolo[1,5-c]pyrimidines to explore the antagonist profiling on adenosine receptors : a preliminary structure-activity relationship study

enthalten in: Journal of medicinal chemistry | 2014

von Federico, S. | Ciancetta, A. | Porta, N. | +6

7

Exploring the directionality of 5-substitutions in a new series of 5-alkylaminopyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine as a strategy to design novel human a(3) adenosine receptor antagonists

enthalten in: Journal of medicinal chemistry | 2012

von Federico, S. | Ciancetta, A. | Sabbadin, D. | +6

8

Exploring potency and selectivity receptor antagonist profiles using a multilabel classification approach : the human adenosine receptors as a key study

enthalten in: Journal of chemical information and modeling | 2009

von Michielan, L. | Stephanie, F. | Terfloth, L. | +6

9

Pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidine derivatives as adenosine receptor antagonists. Influence of the N5 substituent on the affinity at the human A 3 and A 2B adenosine receptor subtypes : a molecular modeling investigation

enthalten in: Journal of medicinal chemistry | 2003

von Pastorin, G. | Da Ros, T. | Spalluto, G. | +7

10

Synthesis, biological properties, and molecular modeling investigation of the first potent, selective, and water-soluble human A(3) adenosine receptor antagonist

enthalten in: Journal of medicinal chemistry | 2002

von Maconi, A. | Pastorin, G. | Da Ros, T. | +8