Suchergebnisse - (Person:"Spalluto, Giampiero")

PubPharm (9)

1

Structure Activity Relationship of 4-Amino-2-thiopyrimidine Derivatives as Platelet Aggregation Inhibitors

enthalten in: Medicinal chemistry (Shariqah (United Arab Emirates)) | 2019

von Cacciari, B. | Crepaldi, P. | Cheng, C. | +5

2

1,2,4]Triazolo[1,5-c]pyrimidines as adenosine receptor antagonists : Modifications at the 8 position to reach selectivity towards A3 adenosine receptor subtype

enthalten in: European journal of medicinal chemistry | 2018

von Federico, S. | Margiotta, E. | Salmaso, V. | +5

3

Discovery of indolylpiperazinylpyrimidines with dual-target profiles at adenosine A2A and dopamine D2 receptors for Parkinson's disease treatment

enthalten in: PloS one | 2018

von Shao, Y. | Ma, X. | Paira, P. | +11

4

Pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidines and Structurally Simplified Analogs. Chemistry and SAR Profile as Adenosine Receptor Antagonists

enthalten in: Current topics in medicinal chemistry | 2016

von Redenti, S. | Ciancetta, A. | Pastorin, G. | +4

5

The Influence of the 1-(3-Trifluoromethyl-Benzyl)-1H-Pyrazole-4-yl Moiety on the Adenosine Receptors Affinity Profile of Pyrazolo[4,3-e][1,2,4]Triazolo[1,5-c]Pyrimidine Derivatives

enthalten in: PloS one | 2015

von Federico, S. | Redenti, S. | Sturlese, M. | +6

6

Scaffold decoration at positions 5 and 8 of 1,2,4-triazolo[1,5-c]pyrimidines to explore the antagonist profiling on adenosine receptors : a preliminary structure-activity relationship study

enthalten in: Journal of medicinal chemistry | 2014

von Federico, S. | Ciancetta, A. | Porta, N. | +6

7

Exploring the directionality of 5-substitutions in a new series of 5-alkylaminopyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine as a strategy to design novel human a(3) adenosine receptor antagonists

enthalten in: Journal of medicinal chemistry | 2012

von Federico, S. | Ciancetta, A. | Sabbadin, D. | +6

8

Pharmacophore elucidation for a new series of 2-aryl-pyrazolo-triazolo-pyrimidines as potent human A3 adenosine receptor antagonists

enthalten in: Bioorganic & medicinal chemistry letters | 2011

von Cheong, S. | Federico, S. | Venkatesan, G. | +5

9

The significance of 2-furyl ring substitution with a 2-(para-substituted) aryl group in a new series of pyrazolo-triazolo-pyrimidines as potent and highly selective hA(3) adenosine receptors antagonists : new insights into structure-affinity relationship and receptor-antagonist recognition

enthalten in: Journal of medicinal chemistry | 2010

von Cheong, S. | Dolzhenko, A. | Kachler, S. | +8

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