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topic_facet:"Poly(ADP-ribose) Polymerase Inhibitors"
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PubPharm (47)
41
Potentiation of cytotoxic drug activity in human tumour cell lines, by amine-substituted 2-arylbenzimidazole-4-carboxamide PARP-1 inhibitors
enthalten in:
Bioorganic & medicinal chemistry letters
| 2004
von
White, A.
|
Curtin, N.
|
Eastman, B.
| +9
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42
Novel poly(ADP-ribose) polymerase-1 inhibitor, AG14361, restores sensitivity to temozolomide in mismatch repair-deficient cells
enthalten in:
Clinical cancer research : an official journal of the American Association for Cancer Research
| 2004
von
Curtin, N.
|
Wang, L.
|
Yiakouvaki, A.
| +8
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43
Anticancer chemosensitization and radiosensitization by the novel poly(ADP-ribose) polymerase-1 inhibitor AG14361
enthalten in:
Journal of the National Cancer Institute
| 2004
von
Calabrese, C.
|
Almassy, R.
|
Barton, S.
| +18
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44
Radiosensitization and DNA repair inhibition by the combined use of novel inhibitors of DNA-dependent protein kinase and poly(ADP-ribose) polymerase-1
enthalten in:
Cancer research
| 2003
von
Veuger, S.
|
Curtin, N.
|
Richardson, C.
| +2
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45
Identification of potent nontoxic poly(ADP-Ribose) polymerase-1 inhibitors : chemopotentiation and pharmacological studies
enthalten in:
Clinical cancer research : an official journal of the American Association for Cancer Research
| 2003
von
Calabrese, C.
|
Batey, M.
|
Thomas, H.
| +12
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46
Tricyclic benzimidazoles as potent poly(ADP-ribose) polymerase-1 inhibitors
enthalten in:
Journal of medicinal chemistry
| 2003
von
Skalitzky, D.
|
Marakovits, J.
|
Maegley, K.
| +12
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47
Novel tricyclic poly(ADP-ribose) polymerase-1 inhibitors with potent anticancer chemopotentiating activity : design, synthesis, and X-ray cocrystal structure
enthalten in:
Journal of medicinal chemistry
| 2002
von
Canan Koch, S.
|
Thoresen, L.
|
Tikhe, J.
| +22
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Thema: Poly(ADP-ribose) Polymerase Inhibitors
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47
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Thema
47
Journal Article
Poly(ADP-ribose) Polymerase Inhibitors
30
Research Support, Non-U.S. Gov't
23
Antineoplastic Agents
22
EC 2.4.2.30
20
Enzyme Inhibitors
19
Poly(ADP-ribose) Polymerases
15
Indoles
12
7GR28W0FJI
12
8237F3U7EH
12
Dacarbazine
12
Temozolomide
12
YF1K15M17Y
12
rucaparib
9
Review
8
12794-10-4
8
Benzodiazepines
8
Poly (ADP-Ribose) Polymerase-1
7
1-(4-dimethylaminomethylphenyl)-8,9-dihydro-7H-...
7
Azulenes
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Erscheinungszeitraum
3
2020-
27
2010-2019
17
2000-2009
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47
Englisch
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