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topic_facet:"Histone Deacetylase Inhibitors"
topic_facet:"Cancer"
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PubPharm (6)
1
Development of decision trees to discriminate HDAC8 inhibitors and non-inhibitors using recursive partitioning
enthalten in:
Journal of biomolecular structure & dynamics
| 2021
von
Amin, S.
|
Adhikari, N.
|
Jha, T.
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2
Histone deacetylase 3 (HDAC3) inhibitors as anticancer agents : A review
enthalten in:
European journal of medicinal chemistry
| 2020
von
Sarkar, R.
|
Banerjee, S.
|
Amin, S.
| +2
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3
Design, synthesis, biological evaluation and molecular docking study of arylcarboxamido piperidine and piperazine-based hydroxamates as potential HDAC8 inhibitors with promising anticancer activity
enthalten in:
European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences
| 2019
von
Trivedi, P.
|
Adhikari, N.
|
Amin, S.
| +4
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4
Histone deacetylase 8 (HDAC8) and its inhibitors with selectivity to other isoforms : An overview
enthalten in:
European journal of medicinal chemistry
| 2019
von
Banerjee, S.
|
Adhikari, N.
|
Amin, S.
| +1
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5
HDAC3 is a potential validated target for cancer : An overview on the benzamide-based selective HDAC3 inhibitors through comparative SAR/QSAR/QAAR approaches
enthalten in:
European journal of medicinal chemistry
| 2018
von
Adhikari, N.
|
Amin, S.
|
Trivedi, P.
| +2
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6
Structure-activity relationships of HDAC8 inhibitors : Non-hydroxamates as anticancer agents
enthalten in:
Pharmacological research
| 2018
von
Amin, S.
|
Adhikari, N.
|
Jha, T.
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1
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Thema: Histone Deacetylase Inhibitors
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Thema: Cancer
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European journal of medicinal chemistry
1
European journal of pharmaceutical sciences : o...
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Journal of biomolecular structure & dynamics
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Cancer
Histone Deacetylase Inhibitors
6
Journal Article
5
EC 3.5.1.98
5
Histone Deacetylases
4
HDAC8 inhibitor
4
Review
3
Antineoplastic Agents
3
HDAC8 protein, human
3
Repressor Proteins
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SAR
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histone deacetylase 3
2
Histone deacetylase
2
Structure-activity relationship (SAR)
1
1RTM4PAL0V
1
67I85E138Y
1
6X80438640
1
Benzamide
1
Benzamides
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Comparative Study
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2020-
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2010-2019
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