Suchergebnisse - (Person:"Spalluto, Giampiero")

PubPharm (183)

71

Synthesis and pharmacological characterization of a new series of 5,7-disubstituted-[1,2,4]triazolo[1,5-a][1,3,5]triazine derivatives as adenosine receptor antagonists: A preliminary inspection of ligand–receptor recognition process

enthalten in: Bioorganic & medicinal chemistry | 2010

von Pastorin, G. | Federico, S. | Paoletta, S. | +8

72

ChemInform Abstract: Comparison of Nine Programs Predicting pKa Values of Pharmaceutical Substances.

enthalten in: ChemInform | 2010

von Michielan, L. | Stephanie, F. | Terfloth, L. | +6

73

Receptor-driven identification of novel human A₃ adenosine receptor antagonists as potential therapeutic agents

enthalten in: Methods in enzymology | 2010

von Paoletta, S. | Federico, S. | Spalluto, G. | +1

74

13 Receptor-Driven Identification of Novel Human A3 Adenosine Receptor Antagonists as Potential Therapeutic Agents

enthalten in: Methods in enzymology | 2010

von Paoletta, S. | Federico, S. | Spalluto, G. | +1

75

GPU Accelerated Support Vector Machines for Mining High-Throughput Screening Data

enthalten in: Journal of chemical information and modeling | 2009

von Michielan, L. | Stephanie, F. | Terfloth, L. | +6

76

Exploring potency and selectivity receptor antagonist profiles using a multilabel classification approach : the human adenosine receptors as a key study

enthalten in: Journal of chemical information and modeling | 2009

von Michielan, L. | Stephanie, F. | Terfloth, L. | +6

77

Combining selectivity and affinity predictions using an integrated Support Vector Machine (SVM) approach : An alternative tool to discriminate between the human adenosine A(2A) and A(3) receptor pyrazolo-triazolo-pyrimidine antagonists binding sites

enthalten in: Bioorganic & medicinal chemistry | 2009

von Michielan, L. | Bolcato, C. | Federico, S. | +9

78

6-Amino-2-mercapto-3H-pyrimidin-4-one derivatives as new candidates for the antagonism at the P2Y12 receptors

enthalten in: Bioorganic & medicinal chemistry | 2009

von Crepaldi, P. | Cacciari, B. | Bonache, M. | +8

79

Human A3 adenosine receptor as versatile G protein-coupled receptor example to validate the receptor homology modeling technology

enthalten in: Current pharmaceutical design | 2009

von Morizzo, E. | Federico, S. | Spalluto, G. | +1

80

6-Amino-2-mercapto-3H-pyrimidin-4-one derivatives as new candidates for the antagonism at the P2Y12 receptors

enthalten in: Bioorganic & medicinal chemistry | 2009

von Crepaldi, P. | Cacciari, B. | Bonache, M. | +8