Suchergebnisse - (Person:"Spalluto, Giampiero")

PubPharm (11)

1

1,2,4]Triazolo[1,5-c]pyrimidines as Tools to Investigate A3 Adenosine Receptors in Cancer Cell Lines

enthalten in: ChemMedChem | 2023

von Federico, S. | Persico, M. | Trevisan, L. | +11

2

Design, Synthesis and Evaluation of New Indolylpyrimidylpiperazines for Gastrointestinal Cancer Therapy

enthalten in: Molecules (Basel, Switzerland) | 2019

von Tan, A. | Babak, M. | Venkatesan, G. | +10

3

A2A Adenosine Receptor Antagonists as Therapeutic Candidates : Are They Still an Interesting Challenge?

enthalten in: Mini reviews in medicinal chemistry | 2018

von Cacciari, B. | Spalluto, G. | Federico, S.

4

Discovery of indolylpiperazinylpyrimidines with dual-target profiles at adenosine A2A and dopamine D2 receptors for Parkinson's disease treatment

enthalten in: PloS one | 2018

von Shao, Y. | Ma, X. | Paira, P. | +11

5

Scaffold decoration at positions 5 and 8 of 1,2,4-triazolo[1,5-c]pyrimidines to explore the antagonist profiling on adenosine receptors : a preliminary structure-activity relationship study

enthalten in: Journal of medicinal chemistry | 2014

von Federico, S. | Ciancetta, A. | Porta, N. | +6

6

Revisiting a receptor-based pharmacophore hypothesis for human A(2A) adenosine receptor antagonists

enthalten in: Journal of chemical information and modeling | 2013

von Bacilieri, M. | Ciancetta, A. | Paoletta, S. | +9

7

8-(2-Furyl)adenine derivatives as A₂A adenosine receptor ligands

enthalten in: European journal of medicinal chemistry | 2013

von Dal Ben, D. | Buccioni, M. | Lambertucci, C. | +6

8

Combining selectivity and affinity predictions using an integrated Support Vector Machine (SVM) approach : An alternative tool to discriminate between the human adenosine A(2A) and A(3) receptor pyrazolo-triazolo-pyrimidine antagonists binding sites

enthalten in: Bioorganic & medicinal chemistry | 2009

von Michielan, L. | Bolcato, C. | Federico, S. | +9

9

Linear and nonlinear 3D-QSAR approaches in tandem with ligand-based homology modeling as a computational strategy to depict the pyrazolo-triazolo-pyrimidine antagonists binding site of the human adenosine A2A receptor

enthalten in: Journal of chemical information and modeling | 2008

von Michielan, L. | Bacilieri, M. | Schiesaro, A. | +7

10

Medicinal chemistry of A2A adenosine receptor antagonists

enthalten in: Current topics in medicinal chemistry | 2003

von Cacciari, B. | Pastorin, G. | Spalluto, G.