Atogepant for migraine

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Atogepant is a selective oral, small-molecule calcitonin gene-related peptide (CGRP) receptor antagonist that has been approved for preventive treatment of migraine. CGRP is a neuropeptide involved in vasodilation and cerebrovascular regulation. CGRP is the most potent vasoactive constituent of the cerebrovascular trigeminal neuronal system and has a key role in migraine. Medications targeting CGRP are being used as migraine preventive and abortive treatments.

Medienart:

E-Artikel

Erscheinungsjahr:

2022

Erschienen:

2022

Enthalten in:

Zur Gesamtaufnahme - volume:58

Enthalten in:

Drugs of today (Barcelona, Spain : 1998) - 58(2022), 8 vom: 19. Aug., Seite 399-405

Sprache:

Englisch

Beteiligte Personen:

Bedrin, Kate [VerfasserIn]
Ailani, Jessica [VerfasserIn]

Links:

Volltext

Themen:

7CRV8RR151
Analgesic drugs
Analgesics
Antimigraine drugs
Atogepant
Calcitonin Gene-Related Peptide
Calcitonin Gene-Related Peptide Receptor Antagonists
Calcitonin gene-related peptide (CGRP) receptor antagonists
Gepants
JHB2QIZ69Z
Journal Article
Migraine with aura
Migraine without aura
Piperidines
Pyridines
Pyrroles
Spiro Compounds

Anmerkungen:

Date Completed 22.08.2022

Date Revised 22.08.2022

published: Print

Citation Status MEDLINE

doi:

10.1358/dot.2022.58.8.3408815

funding:

Förderinstitution / Projekttitel:

PPN (Katalog-ID):

NLM345024966