PYRIMIDINEDIAMINE KINASE INHIBITORS
【課題】ポロ様キナーゼ１（ＰＬＫ１）の活性を含む、キナーゼ活性を阻害するために有用なピリミジンジアミン化合物の提供。【解決手段】式（Ｉ）で示される化合物又は薬学的に許容される塩、溶媒和物、Ｎ−酸化物、又はプロドラッグ。［Ｙ１はＯ又はＳ；Ｚ１はＣＨ又はＮ；Ａはフェニル又は６員のヘテロアリール；Ｒ１〜Ｒ１０はＨ等］【選択図】なし.
| Medienart: |
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Patent| Erscheinungsjahr: |
2015 |
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| Erschienen: |
2015 |
| Enthalten in: |
Europäisches Patentamt - (2015) vom: 27. Aug. Zur Gesamtaufnahme - year:2015 |
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| Sprache: |
Japanisch |
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| Beteiligte Personen: |
RAJINDER SINGH [VerfasserIn] |
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| Links: |
Volltext [kostenfrei] |
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| Anmerkungen: |
Source: www.epo.org (no modifications made), First posted: 2015-08-27, Last update posted on www.tib.eu: 2022-05-22, Last updated: 2023-02-09 |
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| Patentnummer: |
JP2015155447 |
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| Förderinstitution / Projekttitel: |
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| PPN (Katalog-ID): |
EPA012316962 |
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| 520 | |a 【課題】ポロ様キナーゼ１（ＰＬＫ１）の活性を含む、キナーゼ活性を阻害するために有用なピリミジンジアミン化合物の提供。【解決手段】式（Ｉ）で示される化合物又は薬学的に許容される塩、溶媒和物、Ｎ−酸化物、又はプロドラッグ。［Ｙ１はＯ又はＳ；Ｚ１はＣＨ又はＮ；Ａはフェニル又は６員のヘテロアリール；Ｒ１〜Ｒ１０はＨ等］【選択図】なし | ||
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