一种马铃薯三糖齐墩果酸皂苷衍生物及其制备方法和应用

本发明属于药物化学技术领域,具体涉及一种马铃薯三糖齐墩果酸皂苷衍生物及其制备方法和应用。实验研究发现,本发明提供的马铃薯三糖齐墩果酸皂苷衍生物对新型冠状病毒SARS‑CoV‑2具有显著的抑制作用,可应用于制备治疗新型冠状病毒肺炎药物中;其中,部分马铃薯三糖齐墩果酸皂苷衍生物对新型冠状病毒的抑制效果IC50达到了10μM以下,具有非常好的开发潜力,为治疗新型冠状病毒提供了更多的选择。.

Medienart:

Patent

Erscheinungsjahr:

2021

Erschienen:

2021

Enthalten in:

Europäisches Patentamt - (2021) vom: 24. Dez. Zur Gesamtaufnahme - year:2021

Sprache:

Chinesisch

Links:

Volltext [kostenfrei]

Themen:

615
A61K: Preparations for medical, dental, or toilet purposes (devices or methods specially adapted for bringing pharmaceutical products into particular physical or administering forms a61j0003000000;chemical aspects of, or use of materials for deodorisation of air, for disinfection or sterilisation, or for bandages, dressings, absorbent pads or surgical articles a61l; soap compositions c11d)
A61P: Specific therapeutic activity of chemical compounds or medicinal preparations
C07H: Sugars; derivatives thereof; nucleosides; nucleotides; nucleic acids (derivatives of aldonic or saccharic acids c07c, c07d;aldonic acids, saccharic acids c07c0059105000, c07c0059285000;cyanohydrins c07c0255160000;glycals c07d;compounds of unknown constitution c07g;polysaccharides, derivatives thereof c08b;dna or rna concerning genetic engineering, vectors, e.g. plasmids, or their isolation, preparation or purification c12n0015000000;sugar industry c13)
C07J: Steroids (seco-steroids c07c)
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Anmerkungen:

Source: www.epo.org (no modifications made), First posted: 2021-12-24, Last update posted on www.tib.eu: 2022-07-13, Last updated: 2023-02-09

Patentnummer:

CN112457363

Förderinstitution / Projekttitel:

PPN (Katalog-ID):

EPA011905441