PYRIMIDONE DERIVATIVES AS SELECTIVE CYTOTOXIC AGENTS AGAINST HIV INFECTED CELLS

The present disclosure is directed to pyrimidone derivatives of Formula I and their use for selectively killing HIV infected GAG-POL expressing cells without concomitant cytotoxicity to HIV nave cells, and for the treatment or prophylaxis of infection by HIV, or for the treatment, prophylaxis or delay in the onset or progression of AIDS or AIDS Related Complex (ARC)..

Medienart:

Patent

Erscheinungsjahr:

2023

Erschienen:

2023

Enthalten in:

Europäisches Patentamt - (2023) vom: 01. Aug. Zur Gesamtaufnahme - year:2023

Sprache:

Englisch

Beteiligte Personen:

CONVERSO ANTONELLA [VerfasserIn]
EL MARROUNI ABDELLATIF [VerfasserIn]
FORSTER ASHLEY [VerfasserIn]
FRIE JESSICA L [VerfasserIn]
HUNTER DAVID N [VerfasserIn]
KUDUK SCOTT D [VerfasserIn]
MITCHELL HELEN J [VerfasserIn]
NANTERMET PHILIPPE [VerfasserIn]
SHA DEYOU [VerfasserIn]
SHIPE WILLIAM DANIEL [VerfasserIn]
WANG CHENG [VerfasserIn]
WANG DEPING [VerfasserIn]

Links:

Volltext [kostenfrei]

Themen:

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Anmerkungen:

Source: www.epo.org (no modifications made), First posted: 2023-08-01, Last update posted on www.tib.eu: 2023-12-04, Last updated: 2023-12-08

Patentnummer:

CA3122571

Förderinstitution / Projekttitel:

PPN (Katalog-ID):

EPA011884444