COMPOUNDS, PHARMACEUTICAL COMPOSITIONS, AND METHODS FOR THE TREATMENT, PREVENTION, OR MANAGEMENT OF HYPERPROLIFERATIVE DISORDER

Disclosed herein are compounds, pharmaceutical compositions, and methods for treating, preventing or managing diseases and conditions including hyperproliferative disorders such as cancer in humans and other mammals. Compounds disclosed herein are PTEFb inhibitor prodrugs, conjugated to an integrin binding moiety via cleavable linkers and/or functional spacers..

Medienart:

Patent

Erscheinungsjahr:

2023

Erschienen:

2023

Enthalten in:

Europäisches Patentamt - (2023) vom: 13. Apr. Zur Gesamtaufnahme - year:2023

Sprache:

Englisch

Beteiligte Personen:

LERCHEN HANS-GEORG [VerfasserIn]
STELTE-LUDWIG BEATRIX [VerfasserIn]
WIEDMANN MAREIKE [VerfasserIn]
LERCHEN ANDREAS [VerfasserIn]
REBSTOCK ANNE-SOPHIE [VerfasserIn]
KOEBBERLING JOHANNES [VerfasserIn]
WONG HARVEY [VerfasserIn]

Links:

Volltext [kostenfrei]

Themen:

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Anmerkungen:

Source: www.epo.org (no modifications made), First posted: 2023-04-13, Last update posted on www.tib.eu: 2023-09-21, Last updated: 2023-09-29

Patentnummer:

WO2023057812

Förderinstitution / Projekttitel:

PPN (Katalog-ID):

EPA002020696