FIBROBLAST ACTIVATION PROTEIN INHIBITOR
Provided are a compound as represented by general formula (I) or a pharmaceutically acceptable salt, a stereoisomer or a solvate thereof, wherein C is a chelator unit; AB is an albumin binding unit; and FAPI is a fibroblast activation protein inhibitor unit. Also provided are a chelate of the above-mentioned compound and a radioactive nuclide, a pharmaceutical composition and the use thereof as a fibroblast activation protein inhibitor for the diagnosis and treatment of diseases.C-AB-FAPI (I).
| Medienart: |
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Patent| Erscheinungsjahr: |
2024 |
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| Erschienen: |
2024 |
| Enthalten in: |
Europäisches Patentamt - (2024) vom: 08. Feb. Zur Gesamtaufnahme - year:2024 |
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| Sprache: |
Englisch |
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| Beteiligte Personen: |
LIU ZHIBO [VerfasserIn] |
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| Links: |
Volltext [kostenfrei] |
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| Themen: |
Sonstige Themen: |
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| Anmerkungen: |
Source: www.epo.org (no modifications made), First posted: 2024-02-08, Last update posted on www.tib.eu: 2024-04-10, Last updated: 2024-04-19 |
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| Patentnummer: |
US2024042066 |
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| Förderinstitution / Projekttitel: |
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| PPN (Katalog-ID): |
EPA00147331X |
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| 520 | |a Provided are a compound as represented by general formula (I) or a pharmaceutically acceptable salt, a stereoisomer or a solvate thereof, wherein C is a chelator unit; AB is an albumin binding unit; and FAPI is a fibroblast activation protein inhibitor unit. Also provided are a chelate of the above-mentioned compound and a radioactive nuclide, a pharmaceutical composition and the use thereof as a fibroblast activation protein inhibitor for the diagnosis and treatment of diseases.C-AB-FAPI (I) | ||
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