Suchergebnisse - (Person:"Maga, Giovanni")

PubPharm (54)

1

New indolylarylsulfone non-nucleoside reverse transcriptase inhibitors show low nanomolar inhibition of single and double HIV-1 mutant strains

enthalten in: European journal of medicinal chemistry | 2020

von Nalli, M. | Armijos Rivera, J. | Masci, D. | +14

2

Chiral Indolylarylsulfone Non-Nucleoside Reverse Transcriptase Inhibitors as New Potent and Broad Spectrum Anti-HIV-1 Agents

enthalten in: Journal of medicinal chemistry | 2017

von Famiglini, V. | La Regina, G. | Coluccia, A. | +14

3

How to win the HIV-1 drug resistance hurdle race : running faster or jumping higher?

enthalten in: The Biochemical journal | 2017

von Garbelli, A. | Riva, V. | Crespan, E. | +1

4

Development and in Vitro Evaluation of a Microbicide Gel Formulation for a Novel Non-Nucleoside Reverse Transcriptase Inhibitor Belonging to the N-Dihydroalkyloxybenzyloxopyrimidines (N-DABOs) Family

enthalten in: Journal of medicinal chemistry | 2016

von Tintori, C. | Brai, A. | Dasso Lang, M. | +14

5

Indolylarylsulfones carrying a heterocyclic tail as very potent and broad spectrum HIV-1 non-nucleoside reverse transcriptase inhibitors

enthalten in: Journal of medicinal chemistry | 2014

von Famiglini, V. | La Regina, G. | Coluccia, A. | +16

6

Exploring the role of 2-chloro-6-fluoro substitution in 2-alkylthio-6-benzyl-5-alkylpyrimidin-4(3H)-ones : effects in HIV-1-infected cells and in HIV-1 reverse transcriptase enzymes

enthalten in: Journal of medicinal chemistry | 2014

von Rotili, D. | Tarantino, D. | Nawrozkij, M. | +12

7

New indolylarylsulfones as highly potent and broad spectrum HIV-1 non-nucleoside reverse transcriptase inhibitors

enthalten in: European journal of medicinal chemistry | 2014

von Famiglini, V. | La Regina, G. | Coluccia, A. | +10

8

New nitrogen containing substituents at the indole-2-carboxamide yield high potent and broad spectrum indolylarylsulfone HIV-1 non-nucleoside reverse transcriptase inhibitors

enthalten in: Journal of medicinal chemistry | 2012

von La Regina, G. | Coluccia, A. | Brancale, A. | +11

9

Synthesis, biological activity, and ADME properties of novel S-DABOs/N-DABOs as HIV reverse transcriptase inhibitors

enthalten in: ChemMedChem | 2012

von Radi, M. | Pagano, M. | Franchi, L. | +11

10

Mechanism of interaction of novel indolylarylsulfone derivatives with K103N and Y181I mutant HIV-1 reverse transcriptase in complex with its substrates

enthalten in: Antiviral chemistry & chemotherapy | 2011

von Samuele, A. | Bisi, S. | Kataropoulou, A. | +5

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