Suchergebnisse - (Person:"Maga, Giovanni")

PubPharm (51)

1

New indolylarylsulfone non-nucleoside reverse transcriptase inhibitors show low nanomolar inhibition of single and double HIV-1 mutant strains

enthalten in: European journal of medicinal chemistry | 2020

von Nalli, M. | Armijos Rivera, J. | Masci, D. | +14

2

Effect of α-Methoxy Substitution on the Anti-HIV Activity of Dihydropyrimidin-4(3 H)-ones

enthalten in: Journal of medicinal chemistry | 2019

von Nawrozkij, M. | Forgione, M. | Yablokov, A. | +16

3

Exploring the role of 2-chloro-6-fluoro substitution in 2-alkylthio-6-benzyl-5-alkylpyrimidin-4(3H)-ones : effects in HIV-1-infected cells and in HIV-1 reverse transcriptase enzymes

enthalten in: Journal of medicinal chemistry | 2014

von Rotili, D. | Tarantino, D. | Nawrozkij, M. | +12

4

New indolylarylsulfones as highly potent and broad spectrum HIV-1 non-nucleoside reverse transcriptase inhibitors

enthalten in: European journal of medicinal chemistry | 2014

von Famiglini, V. | La Regina, G. | Coluccia, A. | +10

5

Mutational analysis of the HIV-1 auxiliary protein Vif identifies independent domains important for the physical and functional interaction with HIV-1 reverse transcriptase

enthalten in: Nucleic acids research | 2014

von Kataropoulou, A. | Bovolenta, C. | Belfiore, A. | +5

ExpressionOfConcernFor: Nucleic Acids Res. 2009 Jun;37(11):3660-9. - PMID 19369217

6

New nitrogen containing substituents at the indole-2-carboxamide yield high potent and broad spectrum indolylarylsulfone HIV-1 non-nucleoside reverse transcriptase inhibitors

enthalten in: Journal of medicinal chemistry | 2012

von La Regina, G. | Coluccia, A. | Brancale, A. | +11

7

2-(Alkyl/aryl)amino-6-benzylpyrimidin-4(3H)-ones as inhibitors of wild-type and mutant HIV-1 : enantioselectivity studies

enthalten in: Journal of medicinal chemistry | 2012

von Rotili, D. | Samuele, A. | Tarantino, D. | +14

8

Mechanism of interaction of novel indolylarylsulfone derivatives with K103N and Y181I mutant HIV-1 reverse transcriptase in complex with its substrates

enthalten in: Antiviral chemistry & chemotherapy | 2011

von Samuele, A. | Bisi, S. | Kataropoulou, A. | +5

9

Enantioselective binding of second generation pyrrolobenzoxazepinones to the catalytic ternary complex of HIV-1 RT wild-type and L100I and K103N drug resistant mutants

enthalten in: Bioorganic & medicinal chemistry letters | 2011

von Butini, S. | Gemma, S. | Brindisi, M. | +11

10

Indolylarylsulfones as HIV-1 non-nucleoside reverse transcriptase inhibitors : new cyclic substituents at indole-2-carboxamide

enthalten in: Journal of medicinal chemistry | 2011

von La Regina, G. | Coluccia, A. | Brancale, A. | +9

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